Oximes: Novel therapeutics with anticancer and anti-inflammatory potential

IA Schepetkin, MB Plotnikov, AI Khlebnikov… - Biomolecules, 2021 - mdpi.com
Oximes have been studied for decades because of their significant roles as
acetylcholinesterase reactivators. Over the last twenty years, a large number of oximes have …

[HTML][HTML] Synthesis and in-silico simulation of some new bis-thiazole derivatives and their preliminary antimicrobial profile: investigation of hydrazonoyl chloride …

RM Kassab, SM Gomha, SA Al-Hussain… - Arabian Journal of …, 2021 - Elsevier
Two new series of bis-thiazoles 6a-f and bis-thiazolones 9a-d were prepared via reacting bis-
thiosemicarbazone 3 with hydrazonoyl chloride derivatives 4a-f and 7a-d, respectively, in …

Synthesis and antimicrobial activity of some new thiazole, thiophene and pyrazole derivatives containing benzothiazole moiety

S Bondock, W Fadaly, MA Metwally - European journal of medicinal …, 2010 - Elsevier
In an attempt to find a new class of antimicrobial agents, a series of thiazole, thiophene,
pyrazole and other related products containing benzothiazole moiety were prepared via the …

Design and synthesis of some thiazolyl and thiadiazolyl derivatives of antipyrine as potential non-acidic anti-inflammatory, analgesic and antimicrobial agents

SAF Rostom, IM El-Ashmawy, HA Abd El Razik… - Bioorganic & medicinal …, 2009 - Elsevier
The synthesis of two groups of structure hybrids comprising basically the antipyrine moiety
attached to either polysubstituted thiazole or 2, 5-disubstituted-1, 3, 4-thiadiazole …

Selective access to 4-substituted 2-aminothiazoles and 4-substituted 5-thiocyano-2-aminothiazoles from vinyl azides and potassium thiocyanate switched by …

B Chen, S Guo, X Guo, G Zhang, Y Yu - Organic letters, 2015 - ACS Publications
A highly selective construction of 4-substituted 2-aminothiazoles and 4-substituted 5-
thiocyano-2-aminothiazoles, respectively, catalyzed by palladium (II) acetate and promoted …

Visible-light-driven synthesis of 4-alkyl/aryl-2-aminothiazoles promoted by in situ generated copper photocatalyst

WL Lei, T Wang, KW Feng, LZ Wu, Q Liu - ACS Catalysis, 2017 - ACS Publications
Room-temperature synthesis of 4-alkyl/aryl-2-aminothiazoles from vinyl azides and
ammonium thiocyanate was accomplished with the aid of copper salts and blue LED …

Synthesis and anti-inflammatory evaluation of some new acyl-hydrazones bearing 2-aryl-thiazole

CM Moldovan, O Oniga, A Parvu, B Tiperciuc… - European journal of …, 2011 - Elsevier
This work describes recent results from our research program aiming at the synthesis and
evaluation of new compounds acting as potential anti-inflammatory drugs. A series of novel …

Synthesis, characterization and in vitro biological activity of mixed transition metal complexes of lornoxicam with 1, 10-phenanthroline

WH Mahmoud, GG Mohamed… - International Journal of …, 2014 - Elsevier
A new series of Cr (III), Mn (II), Fe (II), Fe (III), Co (II), Ni (II) and Zn (II) ternary complexes
derived from lornoxicam and 1, 10-phenanthroline (Phen) have been synthesized and …

Solvent-controlled synthesis of thiocyanated enaminones and 2-aminothiazoles from enaminones, KSCN, and NBS

X Duan, X Liu, X Cuan, L Wang, K Liu… - The Journal of …, 2019 - ACS Publications
An effective and simple solvent-controlled synthesis of thiocyanated enaminones and 2-
aminothiazoles has been demonstrated from enaminones, potassium thiocyanate, and N …

Cyclization of some carbothioamide derivatives containing antipyrine and triazole moieties and investigation of their antimicrobial activities

H Bayrak, A Demirbas, N Demirbas… - European Journal of …, 2010 - Elsevier
Acetohydrazide derivative containing both antipyrine and triazole nuclei (5) was obtained
starting from ethyl hydrazinecarboxylate derivative (2) and 4-aminoantipyrine (1) by three …