The ability of aziridines to undergo highly regio-and stereoselective ring-opening reactions
renders them of great value in organic synthesis. l This ability has not gone unnoticed in …

Vor allem bei enantioselektiven Synthesen werden vicinale Diamine (1, 2‐Diamine) 1 und
Verbindungen, die auf einfachem Weg aus diesen erhalten werden können–wie 1, 2 …

A general, scalable, and highly diastereoselective aziridination of N-tert-butanesulfinyl
ketimino esters is described. The methodology has been utilized to provide straightforward …

This chapter deals with the formation of carbon‐nitrogen bonds by reaction of carbon
nucleophiles with electrophilic aminating reagents. The former encompass aliphatic and …

The synthesis of new nucleoside analogues is currently of high interest. We report here full
details of a study leading to the synthesis of novel isoxazolidinyl analogues of α-amino acid …

N, O-Disubstituted hydroxylamines (R1NHOR2 or NODHA), unlike the O-monosubstituted
derivatives, have received little attention so far. However, they have recently become …

This review covers our recent advances in the synthesis of unusual amino acids in optically
pure form, and their introduction into naturally occurring peptides with specific biological …

A novel organocatalytic approach for aza-Michael reaction of chalcones using commercial
and non-expensive O-benzylhydroxylamine and a readily available organocatalyst is …

Ring Expansion of N-Acyl Aziridine-2-imides to Oxazoline-4-imides, Useful Precursors of
Pure 13-Hydroxy ¢x-Aminoacids. L__/ Page 1 Pergamon Tetrahedron Letters, Vol. 38, No …

In 1999, Bob Atkinson wrote [1] that aziridination reactions were “< qs> epoxidation's poor
relation< qe>”, and this was undoubtedly true at that time: the scope of the synthetic methods …