Further developments and applications of oxazoline-containing ligands in asymmetric catalysis
The chiral oxazoline motif is present in many ligands that have been extensively applied in a
series of important metal-catalyzed enantioselective reactions. This Review aims to provide …
series of important metal-catalyzed enantioselective reactions. This Review aims to provide …
Influenza neuraminidase inhibitors: synthetic approaches, derivatives and biological activity
P Laborda, SY Wang, J Voglmeir - Molecules, 2016 - mdpi.com
Despite being a common viral disease, influenza has very negative consequences, causing
the death of around half a million people each year. A neuraminidase located on the surface …
the death of around half a million people each year. A neuraminidase located on the surface …
Recent Developments in Enantioselective Metal‐Catalyzed Domino Reactions
H Pellissier - Advanced Synthesis & Catalysis, 2016 - Wiley Online Library
This review updates the major progress in the field of enantioselective one‐, two‐, and multi‐
component domino reactions promoted by chiral metal catalysts, covering the literature …
component domino reactions promoted by chiral metal catalysts, covering the literature …
Catalytic asymmetric Friedel–Crafts alkylation of unprotected indoles with nitroalkenes using a novel chiral Yb(OTf)3–pybox complex
Chiral chloro-indeno pybox has served as a new ligand for the Yb (OTf) 3-catalyzed
asymmetric Friedel–Crafts alkylation reaction of indoles with nitroalkenes. The tunable …
asymmetric Friedel–Crafts alkylation reaction of indoles with nitroalkenes. The tunable …
Fast, solvent-free, highly enantioselective three-component coupling of aldehydes, alkynes, and amines catalysed by the copper (II) pybox complex under high …
Z Li, Z Jiang, W Su - Green Chemistry, 2015 - pubs.rsc.org
Chiral propargylamines were synthesized in good to excellent yields with high
enantioselectivity via Cu (OTf) 2/Ph-Pybox catalysed, solvent-free three-component …
enantioselectivity via Cu (OTf) 2/Ph-Pybox catalysed, solvent-free three-component …
The evolution of Tamiflu synthesis, 20 years on: Advent of enabling technologies the last piece of the puzzle?
CR Sagandira, FM Mathe, U Guyo, P Watts - Tetrahedron, 2020 - Elsevier
Influenza is a serious respiratory disease responsible for significant morbidity and mortality
due to both annual epidemics and pandemics; its treatment involves the use of …
due to both annual epidemics and pandemics; its treatment involves the use of …
Asymmetric alkynylation of seven-membered cyclic imines by combining chiral phosphoric acids and Ag (I) catalysts: synthesis of 11-substituted-10, 11 …
YY Ren, YQ Wang, S Liu - The Journal of Organic Chemistry, 2014 - ACS Publications
Asymmetric alkynylation of seven-membered cyclic imine dibenzo [b, f][1, 4] oxazepines is
successfully achieved by combining chiral phosphoric acid and Ag (I) catalysts. Various …
successfully achieved by combining chiral phosphoric acid and Ag (I) catalysts. Various …
Recent advances in the transformations of cycloalkane-fused oxiranes and aziridines
This account highlights the most relevant transformations of cycloalkane-fused oxiranes and
aziridines developed during the past decade with the intention to provide an overview of the …
aziridines developed during the past decade with the intention to provide an overview of the …
Efficient Synthesis of N‐Alkylated 4‐Pyridones by Copper‐Catalyzed Intermolecular Asymmetric Propargylic Amination
Copper‐catalyzed intermolecular asymmetric propargylic amination with 4‐hydroxypyridines
has been realized for the first time. In the presence of Cu complex derived from Pybox …
has been realized for the first time. In the presence of Cu complex derived from Pybox …
Syntheses of natural and biologically relevant products through asymmetric metal-catalyzed domino reactions. A review
H Pellissier - Organic Preparations and Procedures International, 2019 - Taylor & Francis
A challenging goal in synthetic chemistry is the synthesis of complex products from simple
starting materials by using one-step processes such as domino reactions. 1–16 A domino …
starting materials by using one-step processes such as domino reactions. 1–16 A domino …