Coumarins synthesis and transformation via C–H bond activation—a Review

K Szwaczko - Inorganics, 2022 - mdpi.com
For several decades, coumarins have attracted considerable attention due to the fact of their
application in diverse fields such as medical science and biomedical research as well as …

Electrochemical investigation of C-steel corrosion inhibition, in silico, and sulfate-reducing bacteria investigations using pyrazole derivatives

MM Shaban, NM El Basiony, AB Radwan… - ACS …, 2023 - ACS Publications
The inhibitory impact of the two synthesized pyrazole derivatives (3 and 4) toward metallic
and microbial corrosion was investigated. Using open circuit potential, potentiodynamic …

Facile Synthesis of 2‐Methylenebenzothiazoles from Benzothiazole Salts and 4‐Hydroxycoumarins by Ball Milling

S Xu, W Chen, X Yang, J Shi, Z Mai… - Chemistry–An Asian …, 2022 - Wiley Online Library
A simple and practical method for the synthesis of 2‐methylenebenzothiazoles via the
coupling of a benzothiazole salts and 4‐hydroxycoumarins have been described herein …

A short review on the synthesis of oxazolo/thiazolo/imidazolocoumarins and their biological activities

S Patra, P Patra, D Rout, S Adikari… - Synthetic …, 2023 - Taylor & Francis
The coumarins are found in both natural and synthetic compounds that display a broad
spectrum of biological properties including anticoagulant, antibacterial, antioxidant, and …

One-Pot Cascade Access to Ru(II)-Catalyzed Regioselective C(sp2)-H Activation/Alkenylation of Chromeno[4,3-c]pyrazol-4-ones and Their Emission Solvatochromic …

D Singla, K Paul - The Journal of Organic Chemistry, 2022 - ACS Publications
Herein, one-pot cascade synthesis of chromeno [4, 3-c] pyrazol-4-ones and their Ru (II)-
catalyzed regioselective ortho-alkenylation using imine as a weak directing group are done …

Tailoring of novel morpholine-sulphonamide linked thiazole moieties as dual targeting DHFR/DNA gyrase inhibitors: synthesis, antimicrobial and antibiofilm activities …

MM Abdou, EM Eliwa, MAMA Reheim… - New Journal of …, 2024 - pubs.rsc.org
Herein, the chemical synthesis of new thiazole-based benzenesulfonamide-linked
morpholine 4a, b–7via late-stage thiazolation of the corresponding thiosemicarbazone 3 is …

Thiazolation of phenylthiosemicarbazone to access new thiazoles: anticancer activity and molecular docking

WE Elgammal, SS Shaban, EM Eliwa… - Future Medicinal …, 2024 - Taylor & Francis
Aim: Novel thiazole hybrids were synthesized via thiazolation of 4-phenylthiosemicarbazone
(4). Materials & methods: The anticancer activity against the NCI 60 cancer cell line panel …

Non-cytotoxic 3-Acetylcoumarin as an Attractive Target for Human Monoamine Oxidase (HMAO) Enzymes

MO Aghimien, Q Kolawole, PO Igbinoba… - Anticancer …, 2024 - ar.iiarjournals.org
Background/Aim: Coumarins are a broad class of naturally occurring oxygen-heterocyclic
compounds found in plants with diverse biological properties, making them attractive for …

Determining Stable Structure and in Vitro Antiproliferative Properties of a Novel 3‐(2‐((4‐Trifluoromethyl)phenyl)amino)thiazol‐4‐yl)‐2H‐chromen‐2‐one Molecule

A Burak Sarigüney, E Karakaş Sarikaya… - Chemistry & …, 2024 - Wiley Online Library
Since coumarin and thiazole derivatives are known to have antioxidant properties, a novel
derivative was synthesized in this article. 3‐(2‐((4‐(trifluoromethyl) phenyl) amino) thiazol‐4 …

The literature of heterocyclic chemistry, Part XX, 2020

LI Belen'kii, GA Gazieva, YB Evdokimenkova… - Advances in …, 2023 - Elsevier
A systematized survey of reviews and monographs published in 2020 on all aspects of
heterocyclic chemistry is given. Methods for the synthesis, reactivity, and practically useful …