Antifungal drugs: the current armamentarium and development of new agents

N Robbins, GD Wright, LE Cowen - Microbiology spectrum, 2016 - Am Soc Microbiol
Invasive fungal infections are becoming an increasingly important cause of human mortality
and morbidity, particularly for immunocompromised populations. The fungal pathogens …

Functions of sphingolipids in pathogenesis during host–pathogen interactions

J Wang, YL Chen, YK Li, DK Chen, JF He… - Frontiers in …, 2021 - frontiersin.org
Sphingolipids are a class of membrane lipids that serve as vital structural and signaling
bioactive molecules in organisms ranging from yeast to animals. Recent studies have …

Identification of a new class of antifungals targeting the synthesis of fungal sphingolipids

V Mor, A Rella, AM Farnoud, A Singh, M Munshi… - MBio, 2015 - Am Soc Microbiol
Recent estimates suggest that> 300 million people are afflicted by serious fungal infections
worldwide. Current antifungal drugs are static and toxic and/or have a narrow spectrum of …

Sphingolipids as targets for treatment of fungal infections

R Rollin-Pinheiro, A Singh… - Future medicinal …, 2016 - Taylor & Francis
Invasive fungal infections have significantly increased in the last few decades. Three classes
of drugs are commonly used to treat these infections: polyenes, azoles and echinocandins …

Recent progress in the strategic incorporation of fluorine into medicinally active compounds

K Haranahalli, T Honda, I Ojima - Journal of fluorine chemistry, 2019 - Elsevier
This account exemplifies our recent progress on the strategic incorporation of fluorine and
organofluorine groups to (i) taxoid anticancer agents,(ii) acylhydrazone-based antifungal …

Synthesis and biological properties of fungal glucosylceramide

M Del Poeta, L Nimrichter, ML Rodrigues… - PLoS …, 2014 - journals.plos.org
Sphingolipids have recently emerged as key regulators of pathogenicity in a variety of fungi.
Glucosylceramide is a sphingolipid important for fungal cell division, alkaline tolerance …

Old and new strategies in therapy and diagnosis against fungal infections

T Vanzolini, M Magnani - Applied Microbiology and Biotechnology, 2024 - Springer
Fungal infections represent a serious global health threat. The new emerging pathogens
and the spread of different forms of resistance are now hardly challenging the tools available …

[HTML][HTML] Beyond membrane components: uncovering the intriguing world of fungal sphingolipid synthesis and regulation

SA Usmani, M Kumar, K Arya, B Ali, N Bhardwaj… - Research in …, 2023 - Elsevier
Sphingolipids (SLs) are essential to fungal survival and represent a major class of structural
and signaling lipids. Unique SL structures and their biosynthetic enzymes in filamentous …

Methylation of glycosylated sphingolipid modulates membrane lipid topography and pathogenicity of Cryptococcus neoformans

A Singh, H Wang, LC Silva, C Na, M Prieto… - Cellular …, 2012 - Wiley Online Library
In previous studies we showed that the replication of Cryptococcus neoformans in the lung
environment is controlled by the glucosylceramide (GlcCer) synthase gene (GCS1), which …

Vesicular transport systems in fungi

ML Rodrigues, JD Nosanchuk, A Schrank… - Future …, 2011 - Taylor & Francis
Canonical and unconventional mechanisms of secretion in many eukaryotic cells are
relatively well known. In contrast to the situation in animal cells, mechanisms of secretion in …