Beware of docking!

YC Chen - Trends in pharmacological sciences, 2015 - cell.com
Docking is now routine in virtual screening or lead optimization for drug screening and
design. The number of papers related to docking has dramatically increased over the past …

Trends in predictive biodegradation for sustainable mitigation of environmental pollutants: Recent progress and future outlook

AK Singh, M Bilal, HMN Iqbal, A Raj - Science of The Total Environment, 2021 - Elsevier
The feasibility of in-silico techniques, together with the computational framework, has been
applied to predictive bioremediation aiming to clean-up contaminants, toxicity evaluation …

Rosetta FlexPepDock web server—high resolution modeling of peptide–protein interactions

N London, B Raveh, E Cohen, G Fathi… - Nucleic acids …, 2011 - academic.oup.com
Peptide–protein interactions are among the most prevalent and important interactions in the
cell, but a large fraction of those interactions lack detailed structural characterization. The …

Understanding the binding affinity of noscapines with protease of SARS-CoV-2 for COVID-19 using MD simulations at different temperatures

D Kumar, K Kumari, A Jayaraj, V Kumar… - Journal of …, 2021 - Taylor & Francis
The current outbreak of a novel coronavirus, named as SARS-CoV-2 causing COVID-19
occurred in 2019, is in dire need of finding potential therapeutic agents. Recently, ongoing …

Protein-ligand docking in the new millennium–a retrospective of 10 years in the field

SF Sousa, AJM Ribeiro, JTS Coimbra… - Current medicinal …, 2013 - ingentaconnect.com
Protein-ligand docking is currently an important tool in drug discovery efforts and an active
area of research that has been the subject of important developments over the last decade …

[HTML][HTML] Sanjeevini: a freely accessible web-server for target directed lead molecule discovery

B Jayaram, T Singh, G Mukherjee, A Mathur… - BMC …, 2012 - Springer
Background Computational methods utilizing the structural and functional information help
to understand specific molecular recognition events between the target biomolecule and …

SwissDock 2024: major enhancements for small-molecule docking with Attracting Cavities and AutoDock Vina

M Bugnon, UF Röhrig, M Goullieux… - Nucleic Acids …, 2024 - academic.oup.com
Drug discovery aims to identify potential therapeutic compounds capable of modulating the
activity of specific biological targets. Molecular docking can efficiently support this process …

AADS - An Automated Active Site Identification, Docking, and Scoring Protocol for Protein Targets Based on Physicochemical Descriptors

T Singh, D Biswas, B Jayaram - Journal of chemical information …, 2011 - ACS Publications
We report here a robust automated active site detection, docking, and scoring (AADS)
protocol for proteins with known structures. The active site finder identifies all cavities in a …

Promising inhibitors of main protease of novel corona virus to prevent the spread of COVID-19 using docking and molecular dynamics simulation

D Kumar, K Kumari, VK Vishvakarma… - Journal of …, 2021 - Taylor & Francis
Abstract Coronavirus disease-2019 (COVID-19) is a global health emergency and the matter
of serious concern, which has been declared a pandemic by WHO. Till date, no potential …

Discovery of new phenyl sulfonyl-pyrimidine carboxylate derivatives as the potential multi-target drugs with effective anti-Alzheimer's action: Design, synthesis, crystal …

S Manzoor, SK Prajapati, S Majumdar, MK Raza… - European Journal of …, 2021 - Elsevier
Alzheimer's disease (AD) is multifactorial, progressive neurodegeneration with impaired
behavioural and cognitive functions. The multitarget-directed ligand (MTDL) strategies are …