In Silico Computational Studies of Bioactive Secondary Metabolites from Wedelia trilobata against Anti-Apoptotic B-Cell Lymphoma-2 (Bcl-2) Protein Associated with …

HG Gowtham, F Ahmed, S Anandan, CS Shivakumara… - Molecules, 2023 - mdpi.com
In the present study, the binding affinity of 52 bioactive secondary metabolites from Wedelia
trilobata towards the anti-apoptotic B-cell lymphoma-2 (Bcl-2) protein (PDB: 2W3L) structure …

Phytoconstituents of Withania somnifera unveiled Ashwagandhanolide as a potential drug targeting breast cancer: Investigations through computational, molecular …

HG Gowtham, M Murali, SB Singh, C Shivamallu… - Plos one, 2022 - journals.plos.org
Breast cancer is the second most common malignancy in females worldwide and poses a
great challenge that necessitates the identification of novel therapeutic agents from several …

How living cells are affected during the cold atmospheric pressure plasma treatment

F Ghadirian, H Abbasi, O Bavi, A Naeimabadi - Free Radical Biology and …, 2023 - Elsevier
When the electric discharge process is limited by high voltage electrodes shielding, the
ionization measure would be controlled to less than one percent and the temperature to less …

Structure-based screening and validation of bioactive compounds as Zika virus methyltransferase (MTase) inhibitors through first-principle density functional theory …

S Bharadwaj, AK Rao, VD Dwivedi… - Journal of …, 2021 - Taylor & Francis
Recent Zika virus (ZIKV) outbreak and association with human diseases such as
neurological disorders have raised global health concerns. However, in the absence of an …

Luminescence and in-silico studies of binding interactions of arylpiperazinyl-butylbenzoxazolone based synthetic compounds with bovine serum albumin

D Singh, L Kaur, P Singh, A Datta, M Pathak… - … of Photochemistry and …, 2023 - Elsevier
HT 7, a G-protein coupled receptor of CNS is important in regulating various functions of
brain. This study demonstrates the binding interactions of 5-HT specific six synthesized …

Secondary metabolites of Trichoderma spp. as EGFR tyrosine kinase inhibitors: Evaluation of anticancer efficacy through computational approach

HG Gowtham, PD Revanasiddappa, M Murali… - Plos one, 2024 - journals.plos.org
The present study explores the epidermal growth factor receptor (EGFR) tyrosine kinase
inhibition efficacy of secondary metabolites in Trichoderma spp. through molecular docking …

Computational prediction of interaction and pharmacokinetics profile study for polyamino-polycarboxylic ligands on binding with human serum albumin

N Chadha, D Singh, MD Milton, G Mishra… - New Journal of …, 2020 - pubs.rsc.org
Human serum albumin (HSA) is one of the most abundant plasma proteins available in
blood and responsible for transport of fatty acids, drugs and metabolites at its two primary …

Multi-level molecular modelling for plasma medicine

A Bogaerts, N Khosravian, J Van der Paal… - Journal of Physics D …, 2015 - iopscience.iop.org
Modelling at the molecular or atomic scale can be very useful for obtaining a better insight in
plasma medicine. This paper gives an overview of different atomic/molecular scale …

[HTML][HTML] In silico approach to design new cyclooxygenase-2 (COX-2) inhibitors based on MM/QM and ADMET analysis

A Kharwar, A Mishra, VK Singh, AK Tiwari - Chemical Physics Impact, 2024 - Elsevier
In spite of the availability of inhibitors targeting the Cyclooxygenase-2 (COX-2) enzyme,
there persists a need for current medications, not solely within the realm of non-steroidal anti …

Evaluation of potential flavonoid inhibitors of glyoxalase-I based on virtual screening and in vitro studies

A Yadav, R Kumar, A Sunkaria, N Singhal… - Journal of …, 2016 - Taylor & Francis
Glyoxalase-I (GLO-I) is a component of the ubiquitous detoxification system involved in the
conversion of methylglyoxal (MG) to d-lactate in the glycolytic pathway. MG toxicity arises …