Beyond cytotoxic potency: disposition features required to design ADC payload

H Sun, LC Wienkers, A Lee - Xenobiotica, 2024 - Taylor & Francis
Antibody-drug conjugates (ADCs) have demonstrated impressive clinical usefulness in
treating several types of cancer, with the notion of widening of the therapeutic index of the …

An efficient lung cancer detection using optimal SVM and improved weight based beetle swarm optimization

N Venkatesan, S Pasupathy, B Gobinathan - Biomedical Signal Processing …, 2024 - Elsevier
Lung cancer is caused by uncontrolled cell growth in the lung tissue. Early detection of lung
cancer is important for correct detection and availability of treatment. Diagnosing lung …

Targeting urotensin II with silymarin: potential therapeutic strategies for diabetes and associated cardiovascular complications

S Sabarathinam - Phytochemistry Reviews, 2024 - Springer
Diabetes and its associated comorbidities have garnered significant attention in recent
decades, leading to continuous exploration of diagnostic and treatment options. Urotensin II …

[HTML][HTML] Aniline Derivatives Containing 1-Substituted 1, 2, 3-Triazole System as Potential Drug Candidates: Pharmacokinetic Profile Prediction, Lipophilicity Analysis …

E Chrobak, K Bober-Majnusz, M Wyszomirski, A Zięba - Pharmaceuticals, 2024 - mdpi.com
Background: The triazole ring is an attractive structural unit in medicinal chemistry, and
chemical compounds containing this type of system in their structure exhibit a wide spectrum …

Synthesis, Anticancer Activity, and Computational Studies of New Pyrazole Derivatives

AE Khairulah, ZA Shuhaib, RA Alharis… - Russian Journal of …, 2024 - Springer
Abstract new pyrazole derivatives were synthesized through a cyclization reaction of
chalcones derivatives with hydrazine hydrate under acidic catalysis and characterization by …

Sesquiterpene Lactones as Potential G1/S Phase Cell Cycle Inhibitors: A Molecular Docking Study: Sesquiterpene Lactones as Potential Cell Cycle Inhibitors

Z Yousaf, A Zaman, M Ali, M Khan, C Ara… - Pakistan BioMedical …, 2023 - pakistanbmj.com
Cell cycle checkpoints play a crucial role in cell division by monitoring the orderly
progression of each phase, ensuring accurate completion before advancing to the next …

Molecular Docking-Aided Identification of Natural Bioactive Molecules as Potential Cancer Cell Proliferation Inhibitors: Molecular Docking as Cancer Cell Inhibitors

I Hassan, A Zaman, E Zafar, M Khan - Futuristic Biotechnology, 2024 - fbtjournal.com
Cancer is the second leading cause of death worldwide. Uncontrolled proliferation of cells is
a hallmark of cancer development and progression. Ki-67 (a marker of proliferation Kiel-67) …

Identification of Lung Cancer Using Particle Swarm Optimization and Machine Learning Technique

SRR Kabir, H Mondal, A Nag, SMH Jamil… - … Conference on Trends in …, 2023 - Springer
Lung cancer is a specific kind of malignancy that arises in the tissues of the lungs,
specifically in the cells that comprise the lining of the respiratory passages. Smoking is well …