Receptor tyrosine kinase activation: From the ligand perspective

R Trenker, N Jura - Current opinion in cell biology, 2020 - Elsevier
Receptor tyrosine kinases (RTKs) are single-span transmembrane receptors in which
relatively conserved intracellular kinase domains are coupled to divergent extracellular …

Epidermal growth factor receptor: Structure-function informing the design of anticancer therapeutics

RA Mitchell, RB Luwor, AW Burgess - Experimental cell research, 2018 - Elsevier
Research on the epidermal growth factor (EGF) family and the family of receptors (EGFR)
has progressed rapidly in recent times. New crystal structures of the ectodomains with …

Basic Amino Acids Within the Juxtamembrane Domain of the Epidermal Growth Factor Receptor Regulate Receptor Dimerization and Auto-phosphorylation

JD Mohr, A Wagenknecht-Wiesner, DA Holowka… - The protein journal, 2020 - Springer
Epidermal growth factor receptor (EGFR) dysregulation is observed in many human cancers
and is both a cause of oncogenesis and a target for chemotherapy. We previously showed …

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RA Mitchell, RB Luwor, AW Burgess - 2018 - publications.wehi.edu.au
Research on the epidermal growth factor (EGF) family and the family of receptors (EGFR)
has progressed rapidly in recent times. New crystal structures of the ectodomains with …