Triazole hybrid compounds: A new frontier in malaria treatment

L Ravindar, SA Hasbullah, KP Rakesh… - European Journal of …, 2023 - Elsevier
Reviewing the advancements in malaria treatment, the emergence of triazole hybrid
compounds stands out as a groundbreaking development. Combining the advantages of …

Exploring diverse frontiers: Advancements of bioactive 4-aminoquinoline-based molecular hybrids in targeted therapeutics and beyond

L Ravindar, SA Hasbullah, KP Rakesh… - European Journal of …, 2024 - Elsevier
Amongst heterocyclic compounds, quinoline and its derivatives are advantaged scaffolds
that appear as a significant assembly motif for developing new drug entities. Aminoquinoline …

Recent developments in antimalarial activities of 4-aminoquinoline derivatives

L Ravindar, SA Hasbullah, KP Rakesh… - European Journal of …, 2023 - Elsevier
Malaria is the fifth most lethal parasitic infection in the world. Antimalarial medications have
played a crucial role in preventing and eradicating malaria. Numerous heterocyclic moieties …

Metal complexes derived from bidentate ligands: Synthesis, catalytic and biological applications

DI Ugwu, J Conradie - Inorganica Chimica Acta, 2023 - Elsevier
This review focusses on metal complexes containing bidentate ligands. The development in
the synthesis and some applications of these complexes, reported mainly in the last two …

Antimalarial Agents Derived from Metal‐Amodiaquine Complexes with Activity in Multiple Stages of the Plasmodium Life Cycle

L Colina‐Vegas, M da Cruz B. Silva… - … A European Journal, 2023 - Wiley Online Library
Malaria is the one of the deadliest infectious diseases worldwide. Chemically, quinolines are
excellent ligands for metal coordination and are deployed as drugs for malaria treatment …

Antimicrobial Activity of Rhenium Di- and Tricarbonyl Diimine Complexes: Insights on Membrane-Bound S. aureus Protein Binding

K Schindler, Y Cortat, M Nedyalkova, A Crochet… - Pharmaceuticals, 2022 - mdpi.com
Antimicrobial resistance is one of the major human health threats, with significant impacts on
the global economy. Antibiotics are becoming increasingly ineffective as drug-resistance …

Exploring the in vitro anticancer activities of Re (I) picolinic acid and its fluorinated complex derivatives on lung cancer cells: a structural study

ML Matlou, FP Malan, S Nkadimeng, L McGaw… - JBIC Journal of …, 2023 - Springer
Fifteen rhenium (I) tricarbonyl complexes of the form fac-[Re (N, O')(CO) 3 (X)], where N, O'-
bidentate ligand= 2-picolinic acid (Pico); 3, 5-difluoropyridine-2-carboxylic acid (Dfpc); 3 …

Pyridine and Pyrimidine hybrids as privileged scaffolds in antimalarial drug discovery: A recent development

L Ravindar, SA Hasbullah, KP Rakesh… - Bioorganic & Medicinal …, 2024 - Elsevier
Malaria continues to pose a significant threat to global health, which is exacerbated by the
emergence of drug-resistant strains, necessitating the urgent development of new …

Exploring antimalarial potential: Conjugating organometallic moieties with organic fragments for enhanced efficacy

NAZ Norazmi, NH Mukhtar, L Ravindar, AS Saaidin… - Bioorganic …, 2024 - Elsevier
In the search for novel ligands with efficacy against various diseases, particularly parasitic
diseases, molecular hybridization of organometallic units into biologically active scaffolds …

Tricarbonyl rhenium (i) complexes with 8-hydroxyquinolines: structural, chemical, antibacterial, and anticancer characteristics

K Łyczko, A Pogorzelska, U Częścik, M Koronkiewicz… - RSC …, 2024 - pubs.rsc.org
Twelve tricarbonyl rhenium (I) complexes in the '2+ 1'system with the anionic bidentate N, O-
donor ligand (deprotonated 8-hydroxyquinoline (HQ) or its 2-methyl (MeHQ) or 5-chloro …