4-Thiazolidinones: the advances continue…

AC Tripathi, SJ Gupta, GN Fatima, PK Sonar… - European Journal of …, 2014 - Elsevier
The diversity in the biological response of 4-thiazolidinones has attracted the attention of
many researchers to explore this framework for its potential. It is, therefore, of prime …

Novel quinoline/thiazinan-4-one hybrids; design, synthesis, and molecular docking studies as potential anti-bacterial candidates against MRSA

AH Mohamed, SM Mostafa, AA Aly, AA Hassan… - RSC …, 2023 - pubs.rsc.org
In an attempt to develop effective and safe antibacterial agents, we synthesized novel
thiazinanones by combining the quinolone scaffold and the 1, 3-thiazinan-4-one group by …

Transition‐Metal‐Free One‐Pot [3+ 3] Heteroannulative Coupling of Thioamides with Epichlorohydrin: Access to Diverse 1, 3‐Thiazinanes

D Yadav, M Shankar Singh - European Journal of Organic …, 2023 - Wiley Online Library
An operationally simple and efficient cascade approach to access a series of 1, 3‐
thiazinanes has been developed through intermolecular [3+ 3] heteroannulative coupling …

Chemistry of Substituted Thiazinanes and Their Derivatives

AA Hassan, S Bräse, AA Aly, HN Tawfeek - Molecules, 2020 - mdpi.com
Thiazinanes and its isomeric forms represent one of the most important heterocyclic
compounds, and their derivatives represented a highly potent drug in disease treatment …

Bis (benzofuran–thiazolidinone) s and bis (benzofuran–thiazinanone) s as inhibiting agents for chikungunya virus

JR Hwu, NK Gupta, SC Tsay, WC Huang, IC Albulescu… - Antiviral Research, 2017 - Elsevier
There are currently still no approved antiviral drugs to treat or prevent chikungunya virus
(CHIKV) infections despite the fact that this arbovirus continues to cause outbreaks in Africa …

Construction of thiazines and oxathianes via [3+ 3] annulation of N-tosylaziridinedicarboxylates and oxiranes with 1, 4-dithiane-2, 5-diol: application towards the …

RK Varshnaya, P Banerjee - Organic & Biomolecular Chemistry, 2017 - pubs.rsc.org
Lewis acid catalyzed [3+ 3] annulation of N-tosylaziridinedicarboxylates and oxiranes with in
situ generated mercaptoaldehyde for the synthesis of functionalized thiazine and oxathiane …

Convenient diastereoselective synthesis of annulated 3-substituted-(5S*,6S*,Z)-2-(2-(2,4-dinitrophenyl)hydrazono)-5,6-diphenyl-1,3-thiazinan-4-ones

AA Hassan, NK Mohamed, AA Aly, HN Tawfeek… - Molecular Diversity, 2019 - Springer
Abstract Racemic 2-(2, 4-dinitrophenyl) hydrazono)-5, 6-diphenyl-1, 3-thiazinan-4-ones and
(Z)-N′-(2, 4-dinitrophenyl)-2, 3-diphenylacrylohydrazide were formed during the …

[PDF][PDF] Chemistry of 1, 3-thiazin-4-ones and their derivatives, 1995-mid 2018

LJ Silverberg, QJ Moyer - Arkivoc, 2019 - researchgate.net
This review updates an earlier review published in 1996 by Ryabukhin, Korzhavina, and
Suzdalev, which covered the literature through 1994. It deals with the synthesis and …

α/β-Mercaptoalkanoic acids: versatile synthons in the syntheses of fused ring 4-thiazolidinones/thiazolinones/thiazinanones ring system (s)

B Chandrasekhar - Journal of Sulfur Chemistry, 2012 - Taylor & Francis
This review describes the reactions of β-mercaptoalkanoic acids as building blocks for the
synthesis of polyfunctionalized thiazolidinones with pharmacological interest. Annelated …

Facile synthesis of new thiazinanones derived by acenaphythylenone

AA Aly, KU Sadek, MB Alshammari… - Journal of Sulfur …, 2024 - Taylor & Francis
In an attempt to develop new thiazinanones, 2-oxoacenaphthylen-1 (2 H)-ylidene)
hydrazineylidene)-5, 6-diphenyl-1, 3-thiazinan-4-ones were synthesized via the reaction of …