Recent advances in the synthesis of α-amino ketones
Due to the importance of the amino ketone motif in synthetic and medicinal chemistry, the
number of protocols developed in recent years has considerably increased. This review …
number of protocols developed in recent years has considerably increased. This review …
Visible‐light‐driven α‐Oxidation of Amide C(sp3)−H Bonds to Imides via N‐Bromosuccinimide and Water
HH Chang, XX He, ZL Zang, CH Zhou… - Asian Journal of …, 2022 - Wiley Online Library
An efficient, metal‐free oxidation method of the N‐ortho C (sp3)− H bond of amide via visible‐
light irradiation has been developed. A broad range of imides can be facilely obtained at …
light irradiation has been developed. A broad range of imides can be facilely obtained at …
Thiourea-mediated halogenation of alcohols
The halogenation of alcohols under mild conditions expedited by the presence of
substoichiometric amounts of thiourea additives is presented. The amount of thiourea added …
substoichiometric amounts of thiourea additives is presented. The amount of thiourea added …
N-Halosuccinimides as Precatalysts for C-, N-, O-, and X-Nucleophilic Substitution Reactions of Alcohols under Mild Reaction Conditions
N-halosuccinimides (chloro, bromo, and iodo, respectively) were introduced, tested, and
applied as efficient and non-metal precatalysts for C-, N-, O-, and X-nucleophilic substitution …
applied as efficient and non-metal precatalysts for C-, N-, O-, and X-nucleophilic substitution …
NBS-mediated synthesis of β-keto sulfones from benzyl alcohols and sodium arenesulfinates
An efficient synthetic route towards the synthesis of β-keto sulfones has been developed
from secondary benzyl alcohols using N-bromosuccinimide (NBS). The present protocol …
from secondary benzyl alcohols using N-bromosuccinimide (NBS). The present protocol …