Antibacterial and antioxidant activities for natural and synthetic dual-active compounds

G Martelli, D Giacomini - European Journal of Medicinal Chemistry, 2018 - Elsevier
Antimicrobial resistance is widely recognized as a grave threat to global health in the 21st
century, since the past decades have seen a dramatic increase in human-pathogenic …

Transition Metal‐Free Direct Trifluoromethylation of 2,3‐Dihydropyridin‐4(1H)‐ones at Room Temperature

YY Yu, AR Ranade, GI Georg - Advanced Synthesis & Catalysis, 2014 - Wiley Online Library
A transition metal‐free, regioselective C‐5 trifluoromethylation of 2, 3‐dihydropyridin‐4 (1H)‐
ones (cyclic enaminones) with trimethyl (trifluoromethyl) silane (TMSCF3) was developed …

Synthesis of 4-methyl-N′-(3-alkyl-2r, 6c-diarylpiperidin-4-ylidene)-1, 2, 3-thiadiazole-5-carbohydrazides with antioxidant, antitumor and antimicrobial activities

K Paulrasu, A Duraikannu, M Palrasu… - Organic & …, 2014 - pubs.rsc.org
The structures of the newly synthesized 4-methyl-N′-(3-alkyl-2r, 6c-diarylpiperidin-4-
ylidene)-1, 2, 3-thiadiazole-5-carbohydrazide (5a–5l) were confirmed by spectral and …

Aloe Vera Extract‐Mediated CuO NPs as Catalysts for the Synthesis of 4‐Hydroxy‐3‐Methoxybenzaldehyde‐Connected Piperidine Derivatives and Their Antibacterial …

P Packialakshmi, P Gobinath, A Ahamed… - Journal of …, 2023 - Wiley Online Library
We have designed an easy, affordable, and eco‐friendly technique for Schiff base
preparation of vanillin‐coupled piperidine analogues using CuO NPs as a catalyst. Using a …

Ca2+ Ion Sensing by a Piperidin-4-one Derivative and the Effect of β-Cyclodextrin Complexation on the Sensing

M Sumithra, R Sivaraj, GT Selvan… - Journal of …, 2017 - Elsevier
In this paper, we report the turn-on fluorescence based Ca 2+ ion sensing by an anthracene
piperidin-4-one derivative. The compound is obtained using a simple two step synthesis …

Syntheses, characterization and evaluation of novel 2, 6-diarylpiperidin-4-ones as potential analgesic-antipyretic agents

P Tripathi, AC Tripathi, V Chawla, SK Saraf - European Journal of …, 2014 - Elsevier
A novel series of N-(N-methylpiperazinoacetyl)-2, 6-diarylpiperidin-4-one derivatives (1c–3c
and 5c) were synthesized, via base catalyzed nucleophilic substitution of N-chloroacetyl-2, 6 …

[PDF][PDF] BSA Binding, molecular docking and in vitro biological screening of some new 1, 2, 4-triazole heterocycles bearing azinane nucleus

SZ Siddiqui, H Khalid, SJ Laulloo, TA Chohan… - Pak. J. Pharm …, 2020 - researchgate.net
A series of new compounds (5a-q), derived from 5-(1-(4-nitrophenylsulfonyl) piperidin-4-yl)-
4-phenyl-4H-1, 2, 4-triazole-3-thiol (3) were proficiently synthesized to evaluate their …

The Literature of Heterocyclic Chemistry, Part XIII, 2012–2013

LI Belen'kii, YB Evdokimenkova - Advances in Heterocyclic Chemistry, 2015 - Elsevier
A systematized review of reviews and monographs published in 2012–2013 on all aspects
of heterocyclic chemistry is given.

[HTML][HTML] 1, 4, 5-ТРИЗАМЕЩЕННЫЕ 1, 2, 3-ТРИАЗОЛЫ В СИНТЕЗЕ БИИ ПОЛИЦИКЛИЧЕСКИХ СОЕДИНЕНИЙ

ТВ Сокольникова, АГ Пройдаков… - … заведений. Химия и …, 2022 - cyberleninka.ru
В настоящее время азотсодержащие гетероароматические соединения нашли
применение благодаря широкой линейке проявляемой ими биологической активности …

Synthesis, characterization, stereochemistry, antibacterial and antioxidant activity of N-chloroacetyl-2, 6-diphenylpiperidines

S Ponnuswamy, P Chandrika, A Akila, G Usha - Journal of Molecular …, 2023 - Elsevier
A new series of N-chloroacetyl-2, 6-diphenylpiperidines 13–18 have been synthesized from
their corresponding piperidines 7–12. The synthesized compound 14 is unambiguously …