An insight into prodrug strategy for the treatment of Alzheimer's disease

NV Bhilare, VS Marulkar, D Kumar, VK Chatap… - Medicinal Chemistry …, 2022 - Springer
Alzheimer's disease (AD) is the leading cause of dementia worldwide. With 35 million
people over 60 suffering from dementia, new treatments for AD are immediately needed. In …

Glucagon/GLP-1 receptor co-agonists

J Day, J Patterson, J Chabenne, M Dimarchi… - US Patent …, 2013 - Google Patents
First worldwide family litigation filed litigation Critical https://patents. darts-ip. com/? family=
39690775&utm_source= google_patent&utm_medium= platform_link&utm_campaign …

Glucagon analogs exhibiting enhanced solubility and stability in physiological pH buffers

RD DiMarchi, DL Smiley, M Dimarchi… - US Patent …, 2013 - Google Patents
Modified glucagon peptides are disclosed having improved solubility and/or half-life while
retaining glucagon agonist activity. The glycogen peptides have been modified by Sub …

Glucagon analogs exhibiting enhanced solubility in physiological pH buffers

RD DiMarchi, M Dimarchi, J Chabenne - US Patent 8,669,228, 2014 - Google Patents
4,275,152 A 6/1981 Esders et al. 5,359,030 A 10/1994 Ekwuribe(57) ABSTRACT 5,510,459
A 4/1996 Smith et al. 5,512,549 A 4/1996 Chen et a1. Modi? ed glucagon peptides are …

GIP-based mixed agonists for treatment of metabolic disorders and obesity

RD DiMarchi, T Ma - US Patent 9,062,124, 2015 - Google Patents
First worldwide family litigation filed litigation Critical https://patents. darts-ip. com/? family=
41570802&utm_source= google_patent&utm_medium= platform_link&utm_campaign …

Amide based glucagon and superfamily peptide prodrugs

RD DiMarchi, B Kou - US Patent 8,969,288, 2015 - Google Patents
2009-12-18 Assigned to INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY
CORPORATION reassignment INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY …

Glucagon superfamily peptides exhibiting nuclear hormone receptor activity

RD DiMarchi, B Yang, B Finan - US Patent 9,127,088, 2015 - Google Patents
2012-01-09 Assigned to INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY
CORPORATION reassignment INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY …

Glucagon analogs exhibiting physiological solubility and stability

RD DiMarchi, DL Smiley - US Patent 8,338,368, 2012 - Google Patents
4,275,152 A 6, 1981 Esders et al. 5,359,030 A* 10/1994 Ekwuribe..................... 530/303
5,510,459 A* 4, 1996 Smith et al.................... 530/308 5,512,549 A 4, 1996 Chen et …

Glucagon/GLP-1 receptor co-agonists

RD DiMarchi, DL Smiley, M Dimarchi… - US Patent …, 2013 - Google Patents
2009-07-14 Assigned to INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY
CORPORATION reassignment INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY …

Peptide compounds exhibiting glucagon antagonist and GLP-1 agonist activity

RD DiMarchi, B Yang, C Ouyang - US Patent 8,980,830, 2015 - Google Patents
Glucagon analogs are disclosed that exhibit both glucagon antagonist and GLP-1 agonist
activity. In one embodiment, the glucagon antagonist/GLP-1 agonist comprises a modified …