Recent advances in biological active sulfonamide based hybrid compounds Part A: Two-component sulfonamide hybrids

R Ghomashi, S Ghomashi, H Aghaei… - Current Medicinal …, 2023 - ingentaconnect.com
Sulfonamides constitute an important class of drugs, with many types of pharmacological
agents possessing antibacterial, anti-carbonic anhydrase, anti-obesity, diuretic …

Silica supported Brönsted acids as catalyst in organic transformations: A comprehensive review

M Kaur, S Sharma, PMS Bedi - Chinese Journal of Catalysis, 2015 - Elsevier
Brönsted acid catalysts have been used in a number of organic transformations. To
overcome limitations, such as toxicity, volatility, high price and hazardous nature of the …

Electrochemical N-acylation and N-α-ketoacylation of sulfoximines via the selective decarboxylation and dehydration of α-ketoacids

C Kang, M Li, W Huang, S Wang, M Peng, L Zhao… - Green …, 2023 - pubs.rsc.org
Sulfoximines are commonly found in pharmaceuticals, agrochemicals and other biologically
active compounds. However, limited reports exist for their selective functionalization via …

Synthesis and antibacterial activity of sulfonamides. SAR and DFT studies

W Boufas, N Dupont, M Berredjem, K Berrezag… - Journal of Molecular …, 2014 - Elsevier
A series of substituted sulfonamide derivatives were synthesized from chlorosulfonyl
isocyanate (CSI) in tree steps (carbamoylation, sulfamoylation and deprotection) …

[HTML][HTML] Synthesis of some novel coumarin isoxazol sulfonamide hybrid compounds, 3D-QSAR studies, and antibacterial evaluation

SN Esfahani, MS Damavandi, P Sadeghi, Z Nazifi… - Scientific reports, 2021 - nature.com
With the progressive and ever-increasing antibacterial resistance pathway, the need for
novel antibiotic design becomes critical. Sulfonamides are one of the more effective …

[HTML][HTML] Synthesis and anticancer activity assay of novel chalcone-sulfonamide derivatives

APS Bonakdar, F Vafaei, M Farokhpour… - Iranian journal of …, 2017 - ncbi.nlm.nih.gov
Today Cancer remains to be one of the most deadly diseases in the world. Due to the
potential anticancer activity of the chalcone and sulfonamide moieties, five novel hybrid …

Visible-Light-Induced N-Acylation of Sulfoximines

P Qiu, X Duan, M Li, Y Zheng, W Song - Organic Letters, 2022 - ACS Publications
A metal-, base-, and additive-free N-acylation of sulfoximines was developed under mild
conditions using organic photoredox catalyst. This green strategy featured broad substrate …

Influence of dipole moments on the medicinal activities of diverse organic compounds

A Das, A Das, BK Banik - Journal of the Indian Chemical Society, 2021 - Elsevier
In this study, synthesis, biological activity and structure-activity relationships of diverse
compounds are described. In general, the relationships between dipole moment and …

Recent advances in biological active sulfonamide based hybrid compounds part C: Multicomponent sulfonamide hybrids

R Ghomashi, S Ghomashi, H Aghaei… - Current Medicinal …, 2023 - ingentaconnect.com
Sulfonamides, with the general formula R-SO2NR1R2, have attracted great attention since
the early discovery of sulfonamide-containing antibacterial drugs. The combinations of …

Convenient synthesis of novel chalcone and pyrazoline sulfonamide derivatives as potential antibacterial agents

APS Bonakdar, A Sadeghi, HR Aghaei… - Russian Journal of …, 2020 - Springer
Novel chalcone sulfonamide derivatives were synthesized starting from benzophenones
and aldehydes in 3 steps. Also,(E)-3-(4-chlorophenyl)-1-(4-methoxyphenyl) prop-2-en-1-one …