Indole represents one of the most important privileged scaffolds in drug discovery. Indole
derivatives have the unique property of mimicking the structure of peptides and to bind …

Background Various bioactive aromatic compounds containing the indole nucleus showed
clinical and biological applications. Indole scaffold has been found in many of the important …

The iodine catalyzed oxidative system for 3-sulfenylation of indoles with disulfides using
DMSO as oxidant has been achieved under ambient conditions, providing a convenient and …

Due their multifaced applications, the access to organosulfur derivatives in an efficient and
economical way is a challenge in organic synthesis. In this context photochemistry and …

In organic synthesis, transition-metal and photoredox-catalysis-based reaction systems are
emerging trends for the construction of C–S bonds. Many review articles have recently …

Thioyl and sulfonyl radicals are usually produced from various thiols and sulfonyl derivatives
in high efficiency by single-electron-transfer (SET) oxidation. The generated sulfur …

An efficient synthesis of N‐methyl‐3‐chalcogeno‐indoles has been developed via iodine‐
mediated electrophilic annulation reactions of 2‐alkynylaniline derivatives with disulfides or …

An efficient and convenient method was developed for the preparation of 3-sulfenylindoles
via a K2CO3 promoted direct sulfenylation of indoles with disulfides. The method is …

A catalyst-free thiolation of indoles with sulfonyl hydrazides was efficiently developed in
water under mild conditions without any ligand or additive. The reaction provided a variety of …

New indolylarylsulfone derivatives bearing cyclic substituents at indole-2-carboxamide
linked through a methylene/ethylene spacer were potent inhibitors of the WT HIV-1 …