Recent advances in the synthesis of α‐aminophosphonates: A review

A Amira, Z Aouf, H K'tir, Y Chemam… - …, 2021 - Wiley Online Library
Abstract α‐Aminophosphonates play an important role across several fields, including
organic synthesis and various potential applications. This review paper surveys recent …

Design, synthesis and biological evaluation of furan based α-aminophosphonate derivatives as anti-Alzheimer agent

JJ Uparkar, PP Dhavan, BL Jadhav… - Journal of the Iranian …, 2022 - Springer
A series of novel α-aminophosphonates bearing furan motif were designed and were
synthesized under solvent-free condition and further evaluated for inhibition activity of …

[HTML][HTML] Theoretical exploration on structures, bonding aspects and molecular docking of α-aminophosphonate ligated copper complexes against SARS-CoV-2 …

O Yadav, M Kumar, H Mittal, K Yadav… - Frontiers in …, 2022 - frontiersin.org
Recent years have witnessed a growing interest in the biological activity of metal complexes
of α-aminophosphonates. Here for the first time, a detailed DFT study on five α …

[PDF][PDF] Kabachnik–Fields reaction under green conditions—A critical over-view

P Kafarski, MG Górniak, I Andrasiak - Curr. Green Chem., 2015 - researchgate.net
Three-component one-pot Kabachnik-Fields condensation of carbonyl compounds with
amines and phosphites is perhaps the most exploited reaction for the preparation of …

Design, synthesis, cytotoxic evaluation and molecular docking studies of novel thiazolyl α-aminophosphonates

M Gundluru, VN Badavath, HY Shaik, M Sudileti… - Research on Chemical …, 2021 - Springer
A new class of thiazolyl α-aminophosphonate derivatives was synthesized by one-pot
Kabachnik–Fields reaction of ethyl 2-(3-formyl-4-isobutoxyphenyl)-4-methylthiazole-5 …

Microwave-assisted neat synthesis of α-aminophosphonate/phosphinate derivatives of 2-(2-aminophenyl) benzothiazole as potent antimicrobial and antioxidant …

S Thaslim Basha, H Sudhamani… - … , Sulfur, and Silicon …, 2016 - Taylor & Francis
ABSTRACT A series of diethyl/ethylphenyl {2-(benzo [d] thiazol-2-yl) phenylamino}
phosphonates and phosphinates were synthesized under microwave irradiation and neat …

[HTML][HTML] Synthesis and antitumor activity of novel indole derivatives containing α-aminophosphonate moieties

J Ma, J Li, P Guo, X Liao, H Cheng - Arabian Journal of Chemistry, 2021 - Elsevier
A series of novel indole derivatives containing α-aminophosphonate moieties were
synthesized as antitumor agents. The in vitro cytotoxic activity of the compounds was …

Nano Sb2O3 catalyzed green synthesis, cytotoxic activity, and molecular docking study of novel α-aminophosphonates

S Poola, MR Nadiveedhi, S Sarva, M Gundluru… - Medicinal Chemistry …, 2019 - Springer
Green synthesis of a series of novel dialkyl (aryl substituted)(2-fluoro-4-((2-
methylcarbamoyl) pyridine-4-yl) oxy) phenyl) amino) methyl) phosphonates is accomplished …

Green synthesis and anticancer activity of tetrahydrodipyrazolo[3,4‐b:4′,3′‐e]pyridines catalyzed by phospho sulfonic acid

RR Chinthaparthi, VL Chittiboena… - Journal of …, 2021 - Wiley Online Library
Abstract Biologically portent/significant tetrahydrodipyrazolo [3, 4‐b: 4′, 3′‐e] pyridines
are synthesized by an efficient green synthesis of various aldehydes with 3‐methyl‐1 H …

Phosphosulfonic acid‐catalyzed green synthesis and bioassay of α‐aryl‐α‐1,3,4‐thiadiazolyl aminophosphonates

M Gundluru, S Sarva, MKR Kandula… - Heteroatom …, 2016 - Wiley Online Library
A series of new α‐aminophosphonates containing 1, 3, 4‐thiadiazole moiety (4a–l) were
synthesized via a simple, efficient, and one‐pot three‐component Kabachnik–Fields …