Molecular Chaperones of Leishmania: Central Players in Many Stress‐Related and ‐Unrelated Physiological Processes

JM Requena, AM Montalvo… - BioMed research …, 2015 - Wiley Online Library
Molecular chaperones are key components in the maintenance of cellular homeostasis and
survival, not only during stress but also under optimal growth conditions. Folding of nascent …

Systems biology of autophagy in leishmanial infection and its diverse role in precision medicine

V Guhe, P Ingale, A Tambekar, S Singh - Frontiers in Molecular …, 2023 - frontiersin.org
Autophagy is a contentious issue in leishmaniasis and is emerging as a promising
therapeutic regimen. Published research on the impact of autophagic regulation on …

Characterization of the interaction between eupatorin and bovine serum albumin by spectroscopic and molecular modeling methods

H Xu, N Yao, H Xu, T Wang, G Li, Z Li - International Journal of Molecular …, 2013 - mdpi.com
This study investigated the interaction between eupatorin and bovine serum albumin (BSA)
using ultraviolet-visible (UV-vis) absorption, fluorescence, synchronous fluorescence …

Search for Higgs boson decays into pairs of light (pseudo) scalar particles in the γγjj final state in pp collisions at s= 13TeV with the ATLAS detector

M Aaboud, G Aad, B Abbott, B Abeloos, SH Abidi… - Physics Letters B, 2018 - Elsevier
This Letter presents a search for exotic decays of the Higgs boson to a pair of new (pseudo)
scalar particles, H→ aa, where the a particle has a mass in the range 20–60 GeV, and …

Potential Antileukemia Effect and Structural Analyses of SRPK Inhibition by N-(2-(Piperidin-1-yl)-5-(Trifluoromethyl)Phenyl)Isonicotinamide (SRPIN340)

RP Siqueira, ÉAA Barbosa, MD Polêto, GL Righetto… - PloS one, 2015 - journals.plos.org
Dysregulation of pre-mRNA splicing machinery activity has been related to the biogenesis of
several diseases. The serine/arginine-rich protein kinase family (SRPKs) plays a critical role …

Human mitochondrial Hsp70 (mortalin): shedding light on ATPase activity, interaction with adenosine nucleotides, solution structure and domain organization

PR Dores-Silva, LRS Barbosa, CHI Ramos, JC Borges - PloS one, 2015 - journals.plos.org
The human mitochondrial Hsp70, also called mortalin, is of considerable importance for
mitochondria biogenesis and the correct functioning of the cell machinery. In the …

Aspergillus fumigatus Hsp90 interacts with the main components of the cell wall integrity pathway and cooperates in heat shock and cell wall stress adaptation

MC Rocha, K Minari, JHTM Fabri… - Cellular …, 2021 - Wiley Online Library
The initiation of Aspergillus fumigatus infection occurs via dormant conidia deposition into
the airways. Therefore, conidial germination and subsequent hyphal extension and growth …

PtII, PdII and AuIII complexes with a thiosemicarbazone derived from diacethylmonooxime: Structural analysis, trypanocidal activity, cytotoxicity and first insight into the …

ACR Goncalves, ZA Carneiro, CG Oliveira… - European Journal of …, 2017 - Elsevier
New complexes of composition [MX (HL1)](M= Pt II, Pd II, X= Cl− or I−) and [MX (L1)](M= Au
III, X= Cl−; M= Pt II, Pd II, X= PPh 3) have been synthesized using a potentially tridentate …

A docking-based structural analysis of geldanamycin-derived inhibitor binding to human or Leishmania Hsp90

LC Palma, LFGR Ferreira, ALOA Petersen, BRS Dias… - Scientific reports, 2019 - nature.com
Leishmaniasis is a neglected disease that affects millions of individuals around the world.
Regardless of clinical form, treatment is based primarily on the use of pentavalent …

Design, synthesis and in vitro investigation of novel basic celastrol carboxamides as bio-inspired leishmanicidal agents endowed with inhibitory activity against …

I Bassanini, S Parapini, EE Ferrandi, E Gabriele… - Biomolecules, 2021 - mdpi.com
The natural triterpene celastrol (CE) is here used as lead compound for the design and
synthesis of a panel of eleven CE carboxamides that were tested in vitro for their growth …