Strengthening molecular glues: design strategies for improving thalidomide analogs as cereblon effectors and anticancer agents
MJ Nutt, SG Stewart - Drug Discovery Today, 2024 - Elsevier
Highlights•SAR insights on minimum pharmacophore for CRBN binding.•Scaffold alterations
improving drug solubility and stability.•Rational approaches: phenotypic screening, target …
improving drug solubility and stability.•Rational approaches: phenotypic screening, target …
Synthesis and agricultural antimicrobial evaluation of new quinazoline derivatives containing both a piperazine linker and the N‐acetyl moiety
L An, L Yang, T Yan, M Yi, S Liu, H Li… - Pest Management …, 2024 - Wiley Online Library
BACKGROUND To discover more efficient agricultural antimicrobial agents, a series of new
quinazoline derivatives containing both a piperazine linker and the N‐acetyl moiety were …
quinazoline derivatives containing both a piperazine linker and the N‐acetyl moiety were …
[PDF][PDF] An Overview of Antibiotics Used in Cancer Treatment and Drugs that Act as Antimicrotubules
RR Ayyad, AM Mansour, AM Nejm… - Journal of Progress …, 2024 - pioneerpublisher.com
An Overview of Antibiotics Used in Cancer Treatment and Drugs that Act as
Antimicrotubules Page 1 25 An Overview of Antibiotics Used in Cancer Treatment and …
Antimicrotubules Page 1 25 An Overview of Antibiotics Used in Cancer Treatment and …
[PDF][PDF] Beta-1 Receptor (β1) in the Heart Speciic Indicate to Stereoselectivity
RR Ayyad, AM Mansour, AM Nejm, YAA Hassan… - 2024 - pharmacyscijournal.com
The β1 receptor is one of the three beta receptors present in the human body, namely β1,
β2, and β3. The β1 receptor is predominantly located in the heart, where it plays a crucial …
β2, and β3. The β1 receptor is predominantly located in the heart, where it plays a crucial …