From antibacterial to antitumour agents: a brief review on the chemical and medicinal aspects of sulfonamides

H Azevedo-Barbosa, DF Dias, LL Franco… - Mini Reviews in …, 2020 - ingentaconnect.com
Sulfonamides have been in clinical use for many years, and the development of bioactive
substances containing the sulfonamide subunit has grown steadily in view of their important …

Challenges and opportunities: porous supports in carbonic anhydrase immobilization

S Ren, S Jiang, X Yan, R Chen, H Cui - Journal of CO2 Utilization, 2020 - Elsevier
Abstract Carbonic anhydrases (CAs, EC 4.2. 1.1) are zinc-containing metalloenzymes that
can accelerate the hydration rate of CO 2 into HCO 3 _. But natural CA is usually unstable in …

Synthesis of nitrogen, phosphorus, selenium and sulfur-containing heterocyclic compounds–determination of their carbonic anhydrase, acetylcholinesterase …

İ Gülçin, B Trofimov, R Kaya, P Taslimi, L Sobenina… - Bioorganic …, 2020 - Elsevier
Abstract Sulfur-containing pyrroles (1–3), tris (2-pyridyl) phosphine (selenide) sulfide (4–5)
and 4-benzyl-6-(thiophen-2-yl) pyrimidin-2-amine (6) were synthesized and characterized …

Calcium channel blockers: molecular docking and inhibition studies on carbonic anhydrase I and II isoenzymes

C Türkeş, Y Demir, Ş Beydemir - Journal of Biomolecular Structure …, 2021 - Taylor & Francis
Carbonic anhydrases (CAs) are potent dehydration of carbonic acid and catalyst of the
reversible hydration of carbon dioxide. Here, CA I and CA II was purified from human …

Synthesis, characterization, biological evaluation, and in silico studies of novel 1, 3‐diaryltriazene‐substituted sulfathiazole derivatives

M Işık, S Akocak, N Lolak, P Taslimi… - Archiv Der …, 2020 - Wiley Online Library
In the present study, a series of eleven novel 1, 3‐diaryltriazene‐substituted sulfathiazole
moieties (ST1–11) was synthesized by the reaction of diazonium salt of sulfathiazole with …

Synthesis, characterization, molecular docking, and biological activities of coumarin–1, 2, 3‐triazole‐acetamide hybrid derivatives

N Sepehri, M Mohammadi‐Khanaposhtani… - Archiv der …, 2020 - Wiley Online Library
Coumarins and their derivatives are receiving increasing attention due to numerous
biochemical and pharmacological applications. In this study, a series of novel coumarin–1 …

Cholinesterases, α-glycosidase, and carbonic anhydrase inhibition properties of 1H-pyrazolo [1, 2-b] phthalazine-5, 10-dione derivatives: Synthetic analogues for the …

P Taslimi, K Turhan, F Türkan, HS Karaman… - Bioorganic …, 2020 - Elsevier
In this study, using the Cu (OTf) 2 catalyst, 1H-pyrazolo [1, 2-b] phthalazine-5, 10-dione
derivative molecules were carried out in one step and with high yield (86–91%). The …

The synthesis, carbonic anhydrase and acetylcholinesterase inhibition effects of sulfonyl chloride moiety containing oxazolidinones using an intramolecular aza …

A Yıldırım, U Atmaca, E Şahin, P Taslimi… - Journal of …, 2023 - Taylor & Francis
Oxazolidinones are used as various potent antibiotics, in organisms it acts as a protein
synthesis inhibitor, focusing on an initial stage that encompasses the tRNA binding process …

Anticholinergic and antioxidant activities of avocado (Folium perseae) leaves – phytochemical content by LC-MS/MS analysis

L Polat Kose, Z Bingol, R Kaya, AC Goren… - … Journal of Food …, 2020 - Taylor & Francis
In the first stage of the manuscript, we aimed to examine antioxidant capacity and
anticholinergic properties of avocado (Folium perseae) leaves. Avocado leaf was extracted …

Selective hydrodeoxygenation of acetophenone derivatives using a Fe 25 Ru 75@ SILP catalyst: a practical approach to the synthesis of alkyl phenols and anilines

L Goclik, H Walschus, A Bordet, W Leitner - Green Chemistry, 2022 - pubs.rsc.org
A versatile synthetic pathway for the production of valuable alkyl phenols and anilines has
been developed based on the selective hydrodeoxygenation of a wide range of hydroxy …