In consequence of their biological effects, conformationally constrained carbocyclic β-amino
acids have generated great interest among synthetic and medicinal chemists in the past 2 …

Chiral nitrogenated compounds are highly attractive compounds because of their
importance in agrochemicals, fine chemicals, and pharmaceuticals but also due to their …

Peptide-based drug research has received high attention in the field of medicinal chemistry
over the past decade. For drug design, to improve proteolytic stability, it is desirable to …

A straightforward and efficient method for the synthesis of nitrogen‐functionalized
cyclopentane derivatives via [3+ 2] cycloaddition of enamines with donor‐acceptor …

The selective introduction of fluorine onto the skeleton of an aminocyclopentane or
cyclohexane carboxylate has been developed through a novel and efficient fluoride opening …

Abstract Chloramine-T (CAT), the sodium salt of N-chloro-p-toluenesulfonamide, is a low-
cost mild oxidizing agent with a wide range of uses. Most importantly, it can be used in …

Fluorine‐containing organic molecules have generated increasing impact in drug research
over the past decade. Their preparation and development of novel synthetic methods …

This account highlights the most relevant transformations of cycloalkane-fused oxiranes and
aziridines developed during the past decade with the intention to provide an overview of the …

Hydrolytic enzymes, such as lactamases or hydantoinases, can be valuably applied to
convert lactams (cyclic amides) and cyclic imides into optically pure compounds, for …

Organofluorine compounds have had an increasing impact in synthetic organic chemistry
and pharmaceutical research over the past two decades. Their syntheses and the …