Exploration of Synthetic Potential of Quinoline‐3‐Carbaldehydes
Quinoline is one of the most important nitrogen containing heterocycles, being widespread
in nature and present in a broad variety of pharmacologically active compounds …
in nature and present in a broad variety of pharmacologically active compounds …
Chemoselective Intramolecular Morita–Baylis–Hillman Reaction; Acrylamide and Ketone as Sluggish Reacting Partners on a Labile Framework
KC Bharadwaj - The Journal of Organic Chemistry, 2024 - ACS Publications
Chemoselectivity is an important issue frequently encountered while working over labile
precursors. Carbonyl compounds with a heteroatom at the β carbon are sensitive precursors …
precursors. Carbonyl compounds with a heteroatom at the β carbon are sensitive precursors …
Chemoselective and Highly Rate Accelerated Intramolecular Aza-Morita–Baylis–Hillman Reaction
KC Bharadwaj - The Journal of Organic Chemistry, 2018 - ACS Publications
Despite being a very useful C–C bond forming and highly applicative reaction, Morita–Baylis–
Hillman (MBH) reaction has been limited by its excessive slow reaction rate, including its …
Hillman (MBH) reaction has been limited by its excessive slow reaction rate, including its …
Na 2 S-mediated synthesis of terminal alkynes from gem-dibromoalkenes
RM Singh, D Nandini, KC Bharadwaj… - Organic & …, 2017 - pubs.rsc.org
The Na2S-mediated facile synthesis of terminal alkynes from gem-dibromoalkenes, at
20/40° C under open flask conditions has been developed. Various precursors derived from …
20/40° C under open flask conditions has been developed. Various precursors derived from …
Acryl activation by intramolecular hydrogen bond: Morita Baylis Hillman reaction of acrylamide with broad substrate scope
KC Bharadwaj - ChemistrySelect, 2017 - Wiley Online Library
Use of acrylamide as an activated alkene in largely recognized Morita Baylis Hillman (MBH)
reaction has been least explored owing to less reactivity of acrylamide as Michael acceptor …
reaction has been least explored owing to less reactivity of acrylamide as Michael acceptor …
One pot synthesis of 4-iodo-3-phenylbenzo[b][1,6]naphthyridine via imino iodization-cyclization of alkynylquinoline-3-carbaldehydes
R Singh, V Prasad Sharma, R Kumar… - Synthetic …, 2024 - Taylor & Francis
Simple, environmentally benign and metal free one pot strategy has been used for the
synthesis of 4-iodo-3-phenylbenzo [b][1, 6] naphthyridine from O-alkynylquinolinyl …
synthesis of 4-iodo-3-phenylbenzo [b][1, 6] naphthyridine from O-alkynylquinolinyl …
Naphthalenes and Quinolines by Domino Reactions of Morita–Baylis–Hillman Acetates
An efficient synthetic route to highly functionalized naphthalenes and quinolines has been
developed using domino reactions between Morita–Baylis–Hillman (MBH) acetates and …
developed using domino reactions between Morita–Baylis–Hillman (MBH) acetates and …
Dihydroquinolines, dihydronaphthyridines and quinolones by domino reactions of Morita-Baylis-Hillman acetates
An efficient synthetic route to highly substituted dihydroquinolines and
dihydronaphthyridines has been developed using a domino reaction of Morita-Baylis …
dihydronaphthyridines has been developed using a domino reaction of Morita-Baylis …
Facile Metal‐Free Synthesis of Phenanthridines by SN2′ Reaction/C–H Functionalization/Aromatization through the Reaction of Morita–Baylis–Hillman Acetates …
T Gupta, JB Singh, K Mishra, B Maiti… - European Journal of …, 2018 - Wiley Online Library
A simple, highly efficient, and regioselective synthesis of functionalized phenanthridines by
the reaction of MBH acetates of 2‐chloroquinoline‐3‐carbaldehydes with nitroalkanes is …
the reaction of MBH acetates of 2‐chloroquinoline‐3‐carbaldehydes with nitroalkanes is …
Iodine Catalyzed One Pot Synthesis of 4-Iodo-3-Phenylbenzo [B][1, 6] Naphthyridine from Alkynylquinoline-3-Carbaldehydes, Via Imino Iodization of Alkynes
Simple, Metal free, eco-friendly one pot strategy for the synthesis of 4-iodo-3-phenylbenzo
[b][1, 6] naphthyridine is described from O-alkynylquinolinyl aldehydes with tert butyl amine …
[b][1, 6] naphthyridine is described from O-alkynylquinolinyl aldehydes with tert butyl amine …