Antibody-drug conjugates: the new frontier of chemotherapy

S Ponziani, G Di Vittorio, G Pitari, AM Cimini… - International Journal of …, 2020 - mdpi.com
In recent years, antibody-drug conjugates (ADCs) have become promising antitumor agents
to be used as one of the tools in personalized cancer medicine. ADCs are comprised of a …

HER3 in cancer: from the bench to the bedside

L Gandullo-Sánchez, A Ocaña, A Pandiella - Journal of Experimental & …, 2022 - Springer
The HER3 protein, that belongs to the ErbB/HER receptor tyrosine kinase (RTK) family, is
expressed in several types of tumors. That fact, together with the role of HER3 in promoting …

Thirty years of HER3: from basic biology to therapeutic interventions

HM Haikala, PA Jänne - Clinical Cancer Research, 2021 - AACR
HER3 is a pseudokinase member of the EGFR family having a role in both tumor
progression and drug resistance. Although HER3 was discovered more than 30 years ago …

[HTML][HTML] HER3 signaling and targeted therapy in cancer

R Mishra, H Patel, S Alanazi, L Yuan… - Oncology reviews, 2018 - ncbi.nlm.nih.gov
ERBB family members including epidermal growth factor receptor (EGFR) also known as
HER1, ERBB2/HER2/Neu, ERBB3/HER3 and ERBB4/HER4 are aberrantly activated in …

[HTML][HTML] Understanding the biology of HER3 receptor as a therapeutic target in human cancer

H Lyu, A Han, E Polsdofer, S Liu, B Liu - Acta Pharmaceutica Sinica B, 2018 - Elsevier
HER3 belongs to the human epidermal growth factor receptor (HER) family which also
includes HER1/EGFR/erbB1, HER2/erbB2, and HER4/erbB4. As a unique member of the …

Targeting of erbB3 receptor to overcome resistance in cancer treatment

J Ma, H Lyu, J Huang, B Liu - Molecular cancer, 2014 - Springer
The erbB receptors, including the epidermal growth factor receptor (EGFR), erbB2 (also
known as HER2/neu), erbB3 (or HER3), and erbB4 (or HER4), are often aberrantly activated …

Osimertinib and anti-HER3 combination therapy engages immune dependent tumor toxicity via STING activation in trans

JM Vicencio, R Evans, R Green, Z An, J Deng… - Cell Death & …, 2022 - nature.com
Over the past decade, immunotherapy delivered novel treatments for many cancer types.
However, lung cancer still leads cancer mortality, and non-small-cell lung carcinoma …

[HTML][HTML] A comprehensive review of heregulins, HER3, and HER4 as potential therapeutic targets in cancer

JM Mota, KA Collier, RLB Costa, T Taxter, A Kalyan… - Oncotarget, 2017 - ncbi.nlm.nih.gov
Heregulins (HRGs) bind to the receptors HER3 or HER4, induce receptor dimerization, and
trigger downstream signaling that leads to tumor progression and resistance to targeted …

HER-3 surface expression increases in advanced colorectal cancer representing a potential therapeutic target

E Capone, T Tryggvason, I Cela, B Dufrusine… - Cell Death …, 2023 - nature.com
HER-3 (also known as ErbB-3) is a human epidermal growth factor receptor tyrosine kinases
family member, and its expression in CRC (colorectal cancer) tissues was previously …

Emerging anti-cancer antibodies and combination therapies targeting HER3/ERBB3

N Gaborit, M Lindzen, Y Yarden - Human vaccines & …, 2016 - Taylor & Francis
Cancer progression depends on stepwise accumulation of oncogenic mutations and a
select group of growth factors essential for tumor growth, metastasis and angiogenesis …