EGFR mutation mediates resistance to EGFR tyrosine kinase inhibitors in NSCLC: From molecular mechanisms to clinical research

RF Dong, ML Zhu, MM Liu, YT Xu, LL Yuan… - Pharmacological …, 2021 - Elsevier
With the development of precision medicine, molecular targeted therapy has been widely
used in the field of cancer, especially in non-small-cell lung cancer (NSCLC). Epidermal …

[HTML][HTML] Targeted therapies in development for non-small cell lung cancer

T Reungwetwattana, GK Dy - Journal of carcinogenesis, 2013 - ncbi.nlm.nih.gov
The iterative discovery in various malignancies during the past decades that a number of
aberrant tumorigenic processes and signal transduction pathways are mediated by …

Krukovine suppresses KRAS-mutated lung cancer cell growth and proliferation by inhibiting the RAF-ERK pathway and inactivating AKT pathway

H Lai, Y Wang, F Duan, Y Li, Z Jiang, L Luo… - Frontiers in …, 2018 - frontiersin.org
Oncogenic activation of the KRAS gene via point mutations occurs in 20–30% of patients
with non-small cell lung cancer (NSCLC). The RAS-RAF-ERK and RAS-PI3K-AKT pathways …

Prevalence, Clinicopathologic Characteristics, and Molecular Associations of EGFR Exon 20 Insertion Mutations in East Asian Patients with Lung Adenocarcinoma

Y Pan, Y Zhang, Y Li, H Hu, L Wang, H Li… - Annals of surgical …, 2014 - Springer
Purpose To define the prevalence, clinicopathologic characteristics and molecular
associations of epidermal growth factor receptor (EGFR) exon 20 insertion mutations in East …

Drug combinatorial therapies for the treatment of KRAS mutated lung cancers

H He, C Xu, Z Cheng, X Qian… - Current Topics in …, 2019 - ingentaconnect.com
KRAS is the most common oncogene to be mutated in lung cancer, and therapeutics directly
targeting KRAS have proven to be challenging. The mutations of KRAS are associated with …

[HTML][HTML] A novel insertion mutation on exon 20 of epidermal growth factor receptor, conferring resistance to erlotinib

NA Khan, S Mirshahidi, HR Mirshahidi - Case reports in oncology, 2014 - karger.com
The epidermal growth factor receptor (EGFR) is a transmembrane glycoprotein tyrosine
kinase receptor. The small-molecule tyrosine kinase receptor inhibitors (TKIs) are in clinical …