Red blood cells as therapeutic target to treat sickle cell disease

S Bhatt, DA Argueta, K Gupta… - Antioxidants & Redox …, 2024 - liebertpub.com
Significance: Sickle cell disease (SCD) is the most common inherited diathesis affecting
mostly underserved populations globally. SCD is characterized by chronic pain and fatigue …

Modulating hemoglobin allostery for treatment of sickle cell disease: current progress and intellectual property

PP Pagare, A Rastegar, O Abdulmalik… - Expert opinion on …, 2022 - Taylor & Francis
Introduction Sickle cell disease (SCD) is a debilitating inherited disorder that affects millions
worldwide. Four novel SCD therapeutics have been approved, including the hemoglobin …

Isolation and Characterisation of Quercitrin as a Potent Anti-Sickle Cell Anaemia Agent from Alchornea cordifolia

O Adeniyi, R Baptista, S Bhowmick, A Cookson… - Journal of Clinical …, 2022 - mdpi.com
Alchornea cordifolia Müll. Arg.(commonly known as Christmas Bush) has been used
traditionally in Africa to treat sickle cell anaemia (a recessive disease, arising from the S …

Targeted modification of furan‐2‐carboxaldehydes into Michael acceptor analogs yielded long‐acting hemoglobin modulators with dual antisickling activities

AM Omar, O Abdulmalik, KM El‐Say… - Chemical Biology & …, 2024 - Wiley Online Library
Sickle cell disease (SCD) is the most common genetic disorder, affecting millions of people
worldwide. Aromatic aldehydes, which increase the oxygen affinity of human hemoglobin to …

An investigation of structure-activity relationships of azolylacryloyl derivatives yielded potent and long-acting hemoglobin modulators for reversing erythrocyte sickling

AM Omar, O Abdulmalik, MS Ghatge, YA Muhammad… - Biomolecules, 2020 - mdpi.com
Aromatic aldehydes that bind to sickle hemoglobin (HbS) to increase the protein oxygen
affinity and/or directly inhibit HbS polymer formation to prevent the pathological hypoxia …

[PDF][PDF] Isolation and Characterisation of Quercitrin, a Potent Anti-sickle Cell Anaemia Agent from the Nigerian Shrub, Alchornea Spp

OA Adeniyi - 2020 - research.aber.ac.uk
Alchornea spp. is an important plant genus in Africa, where it has been used traditionally by
healers for the treatment of sickle cell anaemia (SCA). SCA is a genetic disorder endemic to …