Recent progress in the development of adenosine receptor ligands as antiinflammatory drugs

R Akkari, JC Burbiel, J Hockemeyer… - Current topics in …, 2006 - ingentaconnect.com
Adenosine receptors belong to the family of G protein-coupled receptors. Four distinct
subtypes are known, termed A1, A2A, A2B and A3. Adenosine is an important signaling …

Structure-based design, synthesis and molecular modeling studies of thiazolyl urea derivatives as novel anti-parkinsonian agents

F Azam, M Vijaya Vara Prasad, N Thangavel… - Medicinal …, 2012 - ingentaconnect.com
Synthesis of 1-(substituted aryl)-3-(thiazol-2-yl) urea derivatives was undertaken as our
efforts to discover novel antiparkinsonian agents with improved pharmacological profile in …

Thiazole compounds and methods of use

S Zhang, A Phadke, C Liu, X Wang, J Quinn… - US Patent …, 2012 - Google Patents
SE A 3. 3. E. 1 compositions containing one or more compounds of Formula eXter et al.
3,933,838 A 1/1976 Manghisi et al. I, or a salt, Solvate, or acylated prodrug of Such …

2-Acylaminothiazole derivative or salt thereof

K Sugasawa, S Watanuki, Y Koga, H Nagata… - US Patent …, 2009 - Google Patents
A 2-acylaminothiazole derivative or a pharmaceutically acceptable salt thereof having an
excellent effect of proliferating human c-mpl-Ba/F3 cells and an activity of increasing …

Method of treating hepatic disease using A2B adenosine receptor antagonists

D Zeng, H Zhong, L Belardinelli - US Patent 7,795,268, 2010 - Google Patents
US7795268B2 - Method of treating hepatic disease using A2B adenosine receptor
antagonists - Google Patents US7795268B2 - Method of treating hepatic disease using A2B …

Azole compound and medicinal use thereof

T Inaba, T Ikemoto, S Sakata, H Maegawa… - US Patent …, 2007 - Google Patents
US7163952B2 - Azole compound and medicinal use thereof - Google Patents
US7163952B2 - Azole compound and medicinal use thereof - Google Patents Azole …

Thiazole derivatives

T Nakajima, M Sugawara, S Uchida, T Ohno… - US Patent …, 2010 - Google Patents
Abstract (Wherein n is an integer of from 0 to 3; R 1 is substituted or unsubstituted cycloalkyl,
substituted or unsubstituted aryl, a substituted or unsubstituted alicyclic heterocyclic group …

Therapeutic and/or preventive agents for a sleep disorder

N Uesaka, S Ichikawa, T Nakajima - US Patent 7,928,098, 2011 - Google Patents
US7928098B2 - Therapeutic and/or preventive agents for a sleep disorder - Google Patents
US7928098B2 - Therapeutic and/or preventive agents for a sleep disorder - Google Patents …

Purine derivatives as agonists of the adenosine A2A receptor

DG Allen, MD Barker, RPC Cousins - US Patent 7,985,740, 2011 - Google Patents
US7985740B2 - Purine derivatives as agonists of the adenosine A2A receptor - Google Patents
US7985740B2 - Purine derivatives as agonists of the adenosine A2A receptor - Google Patents …

Pro-drugs of N-thiazol-2-yl-benzamide derivatives

AG Sams, B Bang-Andersen, G Mikkelsen… - US Patent …, 2010 - Google Patents
DE 855120 C 1, 1953 DE 855120 C 1, 1953 EP 04.07200 A1 1, 1991 EP 870765 A1 10,
1998 EP 0934938 A 8, 1999 EP 1176139 A1 1, 2002 EP 1295872 A1 3, 2003 EP 1354880 …