Fluorine-containing drugs approved by the FDA in 2021

J He, Z Li, G Dhawan, W Zhang, AE Sorochinsky… - Chinese Chemical …, 2023 - Elsevier
Nine new fluorine-containing drugs have been approved by the US Food and Drug
Administration (FDA) in 2021, which are presented in this review article. These small …

Vascular actions of calcitonin gene-related peptide and adrenomedullin

SD Brain, AD Grant - Physiological reviews, 2004 - journals.physiology.org
This review summarizes the receptor-mediated vascular activities of calcitonin gene-related
peptide (CGRP) and the structurally related peptide adrenomedullin (AM). CGRP is a 37 …

ARISE: a phase 3 randomized trial of erenumab for episodic migraine

DW Dodick, M Ashina, JL Brandes, D Kudrow… - …, 2018 - journals.sagepub.com
Background Calcitonin gene-related peptide plays an important role in migraine
pathophysiology. Erenumab, a human monoclonal antibody that inhibits the calcitonin gene …

Safety and efficacy of erenumab for preventive treatment of chronic migraine: a randomised, double-blind, placebo-controlled phase 2 trial

S Tepper, M Ashina, U Reuter, JL Brandes… - The Lancet …, 2017 - thelancet.com
Background The calcitonin gene-related peptide (CGRP) pathway is important in migraine
pathophysiology. We assessed the efficacy and safety of erenumab, a fully human …

Interictal increase of CGRP levels in peripheral blood as a biomarker for chronic migraine

E Cernuda-Morollón, D Larrosa, C Ramón, J Vega… - Neurology, 2013 - AAN Enterprises
Objective: To determine calcitonin gene-related peptide (CGRP) levels outside migraine
attacks in peripheral blood as a potential biomarker for chronic migraine (CM). Methods …

Tension-type headache

S Ashina, DD Mitsikostas, MJ Lee, N Yamani… - Nature Reviews …, 2021 - nature.com
Tension-type headache (TTH) is the most prevalent neurological disorder worldwide and is
characterized by recurrent headaches of mild to moderate intensity, bilateral location …

Neurobiology of migraine

PJ Goadsby, AR Charbit, AP Andreou, S Akerman… - Neuroscience, 2009 - Elsevier
Migraine is a complex disorder of the brain whose mechanisms are only now being
unraveled. It is common, disabling and economically costly. The pain suggests an important …

Tension-type headache: current research and clinical management

A Fumal, J Schoenen - The Lancet Neurology, 2008 - thelancet.com
Tension-type headache (TTH) is the most common form of headache, and chronic tension-
type headache (CTTH) is one of the most neglected and difficult types of headache to treat …

Calcitonin receptor‐like receptor (CLR), receptor activity‐modifying protein 1 (RAMP1), and calcitonin gene‐related peptide (CGRP) immunoreactivity in the rat …

JK Lennerz, V Rühle, EP Ceppa… - Journal of …, 2008 - Wiley Online Library
Calcitonin gene‐related peptide (CGRP) is a key mediator in primary headaches including
migraine. Animal models of meningeal nociception demonstrate both peripheral and central …

OnabotulinumtoxinA decreases interictal CGRP plasma levels in patients with chronic migraine

E Cernuda-Morollón, C Ramón, P Martínez-Camblor… - Pain, 2015 - journals.lww.com
OnabotulinumtoxinA (onabotA) has shown efficacy in chronic migraine (CM). Its mechanism
of action, however, remains obscure. We have analysed whether treatment with onabotA is …