Merging the versatile functionalities of boronic acid with peptides
Y Tan, J Wu, L Song, M Zhang, CJ Hipolito… - International journal of …, 2021 - mdpi.com
Peptides inherently feature the favorable properties of being easily synthesized, water-
soluble, biocompatible, and typically non-toxic. Thus, boronic acid has been widely …
soluble, biocompatible, and typically non-toxic. Thus, boronic acid has been widely …
A boron delivery antibody (BDA) with boronated specific residues: new perspectives in boron neutron capture therapy from an in silico investigation
Boron Neutron Capture Therapy (BNCT) is a tumor cell-selective radiotherapy based on a
nuclear reaction that occurs when the isotope boron-10 (10B) is radiated by low-energy …
nuclear reaction that occurs when the isotope boron-10 (10B) is radiated by low-energy …
Peptide Boronic Acids by Late‐Stage Hydroboration on the Solid Phase
M Werner, J Brinkhofer, L Hammermüller… - Advanced …, 2024 - Wiley Online Library
Organoboron compounds have a wide range of applications in numerous research fields,
and metmhods to incorporate them in biomolecules are much sought after. Here, on‐resin …
and metmhods to incorporate them in biomolecules are much sought after. Here, on‐resin …
Synthesis and Application of Constrained Amidoboronic Acids Using Amphoteric Boron-Containing Building Blocks
Amidoboronic acid-containing peptidomimetics are an important class of scaffolds in
chemistry and drug discovery. Despite increasing interest in boron-based enzyme inhibitors …
chemistry and drug discovery. Despite increasing interest in boron-based enzyme inhibitors …
A tandem process for the synthesis of β-aminoboronic acids from aziridines with haloamine intermediates
S Park, J Koo, W Kim, HG Lee - Chemical Communications, 2022 - pubs.rsc.org
An unprecedented synthetic strategy is devised to generate β-aminoboronic acids from
aziridines via a sequential process involving 1, 2-iodoamine formation and radical borylation …
aziridines via a sequential process involving 1, 2-iodoamine formation and radical borylation …
Synthesis of Fluorinated Aminoalkylboronic Acids from Amphoteric α‐Boryl Aldehydes
Our ongoing search for underdeveloped functional group combinations has brought to light
α‐fluorinated aminoalkylboronic acids, a new class of molecules featuring the B‐CF linkage …
α‐fluorinated aminoalkylboronic acids, a new class of molecules featuring the B‐CF linkage …
Synthesis and applications of aminoboronic acids
V Trudel - 2024 - search.proquest.com
Boronic acids are a class of compounds with a wide range of applications enabled by the
coordinative ability of the boron atom. The development of new synthetic methods to access …
coordinative ability of the boron atom. The development of new synthetic methods to access …