Advances in 2H-azirine chemistry: A seven-year update

AF Khlebnikov, MS Novikov, NV Rostovskii - Tetrahedron, 2019 - Elsevier
Abstract 2H-Azirines are versatile building blocks for the preparation of various nitrogen-
containing heterocycles. Seven years ago the comprehensive review on azirine chemistry …

Visible light-assisted chemistry of vinyl azides and its applications in organic synthesis

B Saxena, RI Patel, J Tripathi, A Sharma - Organic & Biomolecular …, 2023 - pubs.rsc.org
Vinyl azides have emerged as highly versatile precursors in organic synthesis due to their
rich reactivity driven by the excellent leaving-group ability of molecular nitrogen. Over the …

Pyrazolo-benzothiazole hybrids: Synthesis, anticancer properties and evaluation of antiangiogenic activity using in vitro VEGFR-2 kinase and in vivo transgenic …

VG Reddy, TS Reddy, C Jadala, MS Reddy… - European journal of …, 2019 - Elsevier
A series of new pyrazolo-benzothiazole hybrids (7–26) were synthesised and screened for
their cytotoxic activity towards several cancer cell lines [colon (HT-29), prostate (PC-3), lung …

Visible-Light-Induced Deaminative Alkylation/Cyclization of Alkyl Amines with N-Methacryloyl-2-phenylbenzoimidazoles in Continuous-Flow Organo-Photocatalysis

V Ramesh, M Gangadhar, JB Nanubolu… - The Journal of Organic …, 2021 - ACS Publications
Herein, we present a metal-free visible-light-induced eosin-y-catalyzed deaminative strategy
for the sequential alkylation/cyclization of N-methacryloyl-2-phenylbenzoimidazoles with …

Synthesis of Imidazo[1,2-a]pyridines via Near UV Light-Induced Cyclization of Azirinylpyridinium Salts

IP Filippov, AV Agafonova, GD Titov… - The Journal of …, 2022 - ACS Publications
An efficient one-pot synthesis of imidazo [1, 2-a] pyridines from 2-bromoazirines and
pyridines has been developed. The construction of the bicyclic framework of imidazo [1, 2-a] …

[HTML][HTML] Recent developments in the photochemical synthesis of functionalized imidazopyridines

C Tran, A Hamze - Molecules, 2022 - mdpi.com
Imidazopyridines constitute one of the most important scaffolds in medicinal chemistry, as
their skeleton could be found in a myriad of biologically active molecules. Although …

Recent Advances on α‐Azidoketones and Esters in the Synthesis of N‐Heterocycles

L Borkotoky, RA Maurya - Asian Journal of Organic Chemistry, 2022 - Wiley Online Library
Organic azides have been proven to possess versatile reactivity that is utilized to synthesize
a large number of molecular scaffolds. Among the azides, α‐azidoketones and esters have …

2H-Azirines as C–C Annulation Reagents in Cu-Catalyzed Synthesis of Furo[3,2-c]quinolone Derivatives

PA Sakharov, NV Rostovskii, AF Khlebnikov… - Organic …, 2019 - ACS Publications
A method of furo-annulation of 4-hydroxy-2-oxoquinoline-3-carboxylates with 3-arylazirines
under Cu (II) catalysis was developed to synthesize a variety of 2, 3-dihydrofuro [3, 2-c] …

Organo‐photocatalytic Synthesis of 6‐β‐Disubstituted Phenanthridines from α‐Diazo‐β‐Keto Compounds and Vinyl Azides

L Devi, A Pokhriyal, S Shekhar, R Kant… - Asian Journal of …, 2021 - Wiley Online Library
An efficient organo‐photocatalytic method for the synthesis of 6‐β‐disubstituted
phenanthridines has been developed. The reaction documents unprecedented generation …

Visible light-promoted [3+ 2] cyclization reaction of vinyl azides with perfluoroalkyl-substituted-imidoyl sulfoxonium ylides

M Yang, YX Meng, H Mehfooz, YL Zhao - Chemical Communications, 2024 - pubs.rsc.org
Visible-light-induced [3+ 2] cyclization of vinyl azides with perfluoroalkyl-substituted imidoyl
sulfoxonium ylides has been developed for the first time. In this transformation, perfluoroalkyl …