Advances in 2H-azirine chemistry: A seven-year update
Abstract 2H-Azirines are versatile building blocks for the preparation of various nitrogen-
containing heterocycles. Seven years ago the comprehensive review on azirine chemistry …
containing heterocycles. Seven years ago the comprehensive review on azirine chemistry …
Visible light-assisted chemistry of vinyl azides and its applications in organic synthesis
Vinyl azides have emerged as highly versatile precursors in organic synthesis due to their
rich reactivity driven by the excellent leaving-group ability of molecular nitrogen. Over the …
rich reactivity driven by the excellent leaving-group ability of molecular nitrogen. Over the …
Pyrazolo-benzothiazole hybrids: Synthesis, anticancer properties and evaluation of antiangiogenic activity using in vitro VEGFR-2 kinase and in vivo transgenic …
A series of new pyrazolo-benzothiazole hybrids (7–26) were synthesised and screened for
their cytotoxic activity towards several cancer cell lines [colon (HT-29), prostate (PC-3), lung …
their cytotoxic activity towards several cancer cell lines [colon (HT-29), prostate (PC-3), lung …
Visible-Light-Induced Deaminative Alkylation/Cyclization of Alkyl Amines with N-Methacryloyl-2-phenylbenzoimidazoles in Continuous-Flow Organo-Photocatalysis
V Ramesh, M Gangadhar, JB Nanubolu… - The Journal of Organic …, 2021 - ACS Publications
Herein, we present a metal-free visible-light-induced eosin-y-catalyzed deaminative strategy
for the sequential alkylation/cyclization of N-methacryloyl-2-phenylbenzoimidazoles with …
for the sequential alkylation/cyclization of N-methacryloyl-2-phenylbenzoimidazoles with …
Synthesis of Imidazo[1,2-a]pyridines via Near UV Light-Induced Cyclization of Azirinylpyridinium Salts
IP Filippov, AV Agafonova, GD Titov… - The Journal of …, 2022 - ACS Publications
An efficient one-pot synthesis of imidazo [1, 2-a] pyridines from 2-bromoazirines and
pyridines has been developed. The construction of the bicyclic framework of imidazo [1, 2-a] …
pyridines has been developed. The construction of the bicyclic framework of imidazo [1, 2-a] …
[HTML][HTML] Recent developments in the photochemical synthesis of functionalized imidazopyridines
C Tran, A Hamze - Molecules, 2022 - mdpi.com
Imidazopyridines constitute one of the most important scaffolds in medicinal chemistry, as
their skeleton could be found in a myriad of biologically active molecules. Although …
their skeleton could be found in a myriad of biologically active molecules. Although …
Recent Advances on α‐Azidoketones and Esters in the Synthesis of N‐Heterocycles
L Borkotoky, RA Maurya - Asian Journal of Organic Chemistry, 2022 - Wiley Online Library
Organic azides have been proven to possess versatile reactivity that is utilized to synthesize
a large number of molecular scaffolds. Among the azides, α‐azidoketones and esters have …
a large number of molecular scaffolds. Among the azides, α‐azidoketones and esters have …
2H-Azirines as C–C Annulation Reagents in Cu-Catalyzed Synthesis of Furo[3,2-c]quinolone Derivatives
PA Sakharov, NV Rostovskii, AF Khlebnikov… - Organic …, 2019 - ACS Publications
A method of furo-annulation of 4-hydroxy-2-oxoquinoline-3-carboxylates with 3-arylazirines
under Cu (II) catalysis was developed to synthesize a variety of 2, 3-dihydrofuro [3, 2-c] …
under Cu (II) catalysis was developed to synthesize a variety of 2, 3-dihydrofuro [3, 2-c] …
Organo‐photocatalytic Synthesis of 6‐β‐Disubstituted Phenanthridines from α‐Diazo‐β‐Keto Compounds and Vinyl Azides
An efficient organo‐photocatalytic method for the synthesis of 6‐β‐disubstituted
phenanthridines has been developed. The reaction documents unprecedented generation …
phenanthridines has been developed. The reaction documents unprecedented generation …
Visible light-promoted [3+ 2] cyclization reaction of vinyl azides with perfluoroalkyl-substituted-imidoyl sulfoxonium ylides
M Yang, YX Meng, H Mehfooz, YL Zhao - Chemical Communications, 2024 - pubs.rsc.org
Visible-light-induced [3+ 2] cyclization of vinyl azides with perfluoroalkyl-substituted imidoyl
sulfoxonium ylides has been developed for the first time. In this transformation, perfluoroalkyl …
sulfoxonium ylides has been developed for the first time. In this transformation, perfluoroalkyl …