100 years of the Wolff rearrangement

W Kirmse - European Journal of Organic Chemistry, 2002 - Wiley Online Library
The conversion of α‐diazo ketones into ketenes, and products derived therefrom, was
discovered by Wolff in 1902. Major applications of the Wolff rearrangement, such as the …

Base‐catalyzed hydroamination of olefins: an environmentally friendly route to amines

J Seayad, A Tillack, CG Hartung… - Advanced Synthesis & …, 2002 - Wiley Online Library
The base‐catalyzed hydroamination of olefins offers a simple and elegant access to various
primary, secondary, and tertiary amines. Particular focus is placed on developments in the …

C-glycosides and aza-C-glycosides as potential glycosidase and glycosyltransferase inhibitors

W Zou - Current topics in medicinal chemistry, 2005 - ingentaconnect.com
Glycosylation as one of most important post-translational modification of gene products is
often critical to specific cellular biological functions. Since elevated glycoprocessing enzyme …

Synthesis and bioevaluation of glycosyl ureas as α-glucosidase inhibitors and their effect on mycobacterium

N Tewari, VK Tiwari, RC Mishra, RP Tripathi… - Bioorganic & medicinal …, 2003 - Elsevier
Glycosyl amino esters (2–13) on reaction with different isocyanates resulted in quantitative
conversion to glycosyl ureas (14-–32). Few of the selected ureas (15–20, 22–28, 30 and 32) …

Efficient synthesis of 3-substituted indoles through a domino gold (I) chloride catalyzed cycloisomerization/C3-functionalization of 2-(alkynyl) anilines

C Praveen, K Karthikeyan, PT Perumal - Tetrahedron, 2009 - Elsevier
An efficient synthesis of 3-substituted indoles by a sequential approach involving gold (I)
chloride catalyzed cycloisomerization/bis-addition and conjugate addition of 2-(alkynyl) …

General methods for iminosugar synthesis

L Cipolla, B La Ferla, F Nicotra - Current Topics in Medicinal …, 2003 - ingentaconnect.com
Recent iminosugar syntheses starting both from commercially available sugars and non-
glycidic precursors, are reported in this article. Exploiting carbohydrate starting materials …

Tetra-n-butylammonium fluoride: an efficient base for aza-Michael addition—synthesis of glycosyl β-amino acid esters

GVM Sharma, VG Reddy, AS Chander… - Tetrahedron: Asymmetry, 2002 - Elsevier
Tetra-n-butylammonium fluoride: an efficient base for aza-Michael addition—synthesis of
glycosyl β-amino acid esters - ScienceDirect Skip to main contentSkip to article Elsevier logo …

Recent advances in the synthesis of naturally occurring polyhydroxylated alkaloids

H Yoda - Current Organic Chemistry, 2002 - ingentaconnect.com
A major fraction of the organic compounds isolated from nature are comprised of nitrogen,
oxygen, or sulfur heterocycles. Nirogen-containing substances called alkaloids among them …

Synthesis, computational study and glycosidase inhibitory activity of polyhydroxylated conidine alkaloids—a bicyclic iminosugar

SP Sanap, S Ghosh, AM Jabgunde… - Organic & …, 2010 - pubs.rsc.org
New bicyclic conidine iminosugars 1d and 1e were synthesized from D-glucose. Thus, D-
glucose was converted to sugar β-amino acids 3a and 3b in good yields. Individual …

α-Geminal dihydroxymethyl piperidine and pyrrolidine iminosugars: synthesis, conformational analysis, glycosidase inhibitory activity, and molecular docking studies

NJ Pawar, VS Parihar, ST Chavan… - The Journal of …, 2012 - ACS Publications
The Jocic–Reeve and Corey–Link type reaction of dichloromethyllithium with suitably
protected 5-keto-hexofuranoses followed by treatment with sodium azide and sodium …