Aminoalcohols have been used extensively in asymmetric synthesis, both as chiral ligands
and auxiliaries. The two heteroatoms allow great flexibility, as one or both can be bound to a …

Derivatives of 7-oxabicyclo [2.2. l] heptanes (7-oxanorbornanes) are found in Nature, some
of these having interesting biological activities. Analogues of these compounds have also …

The published data on the intramolecular Diels–Alder reaction in compounds of the 2-
alkenylfuran series are generalised. The methods and conditions for the preparation of …

An efficient and versatile one-pot synthesis of 3, 6a-epoxyisoindoles annelated with oxazine,
oxazole, thiazine, thiazole, pyrimidine fragments and with their benzoannelated analogues …

A novel, direct, and high-yielding stereoselective method for enantiopure 1-substituted
tetrahydroisoquinolines (THIQ) is described. The successful approach, which creates the …

Enantioselective conjugate addition of bis (pinacolato) diboron to α, β-unsaturated imines
proceeds smoothly in water in the presence of a chiral copper (II) complex consisting of Cu …

Condensation of (−)-8-benzylaminomenthol with o-phthaldehyde lead to the chiral perhydro-
1, 3-benzoxazine 2 as single diastereoisomer. That compound reacted with different …

The first lipase‐catalyzed domino reaction is described in which the acyl moiety formed
during the enzymatic kinetic resolution of furfuryl alcohols (±)‐3 with a 1‐ethoxyvinyl ester 2 …

IMDA reactions on chiral perhydro-1, 3-benzoxazines, derived from (−)-8-amino menthol,
bearing a styrene substituent at C-2 acting as diene and an acryl amide acting as dienophile …

Aryllithiums prepared by bromine− lithium interchange in chiral 2-(o-bromophenyl)-
substituted perhydro-1, 3-benzoxazines participate in the intramolecular 6-exo …