Recent advances in the application of the Sonogashira method in the synthesis of heterocyclic compounds
MM Heravi, S Sadjadi - Tetrahedron, 2009 - Elsevier
Conclusions In this review, we have presented numerous very useful processes for the
synthesis of heterocycles, which involve palladium-catalyzed coupling followed by …
synthesis of heterocycles, which involve palladium-catalyzed coupling followed by …
Pyrroles and fused pyrroles: synthesis and therapeutic activities
MS Mohamed, SS Fathallah - Mini-Reviews in Organic …, 2014 - ingentaconnect.com
For several decades, interest in pyrrole derivatives increased due to their pharmaceutical
importance, such as antimicrobial, anti-inflammatory, analgesic, anti-tumor, anti-epileptic …
importance, such as antimicrobial, anti-inflammatory, analgesic, anti-tumor, anti-epileptic …
Microwave‐assisted synthesis and evaluation of antimicrobial activity of 3‐{3‐(s‐aryl and s‐heteroaromatic)acryloyl}‐2H‐chromen‐2‐one derivatives
The exploration of potential utilization of microwaves as an energy source for heterocyclic
synthesis was herein investigated using condensation of 3‐acetylcoumarin (1) with aromatic …
synthesis was herein investigated using condensation of 3‐acetylcoumarin (1) with aromatic …
A sequential metal-catalyzed C− N bond formation in the synthesis of 2-amido-indoles
PY Yao, Y Zhang, RP Hsung, K Zhao - Organic letters, 2008 - ACS Publications
A sequential metal-catalyzed C− N bond formation employing ortho-haloaryl acetylenic
bromides is described. The initial amidation is highly selective for Csp− N bond formation …
bromides is described. The initial amidation is highly selective for Csp− N bond formation …
Palladium-catalysed synthesis and transformation of quinolones
VLM Silva, AMS Silva - Molecules, 2019 - mdpi.com
Palladium-catalysed reactions have had a large impact on synthetic organic chemistry and
have found many applications in target-oriented synthesis. Their widespread use in organic …
have found many applications in target-oriented synthesis. Their widespread use in organic …
Applications of palladium dibenzylideneacetone as catalyst in the synthesis of five-membered N-heterocycles
N Kaur - Synthetic Communications, 2019 - Taylor & Francis
A wide variety of biological activities are possessed by N, O, and S containing heterocycles
and recently many reports appeared for the synthesis of these heterocycles. The synthesis of …
and recently many reports appeared for the synthesis of these heterocycles. The synthesis of …
Scale-up of microwave-assisted reactions in a multimode bench-top reactor
D Dallinger, H Lehmann, JD Moseley… - … Process Research & …, 2011 - ACS Publications
An evaluation of a new bench-top microwave batch reactor that uses a single 1 L reaction
vessel is presented. Several microwave-assisted organic reactions have been scaled-up …
vessel is presented. Several microwave-assisted organic reactions have been scaled-up …
Efficient Synthesis of Fluorescent Coumarins and Phosphorous-Containing Coumarin-Type Heterocycles via Palladium Catalyzed Cross-Coupling Reactions
Quantum-chemical calculations on the spectral properties of some aryl substituted 3-
phosphonocoumarins were performed, and the effect of the substituents in the aryl moiety …
phosphonocoumarins were performed, and the effect of the substituents in the aryl moiety …
Efficient synthesis of aminomethylated pyrroloindoles and dipyrrolopyridines via controlled copper-catalyzed domino multicomponent coupling and bis-cyclization
Y Suzuki, Y Ohta, S Oishi, N Fujii… - The Journal of Organic …, 2009 - ACS Publications
Efficient methods for the synthesis of pyrrole-fused indole derivatives via domino copper-
catalyzed multicomponent coupling and bis-cyclization have been developed. The mono-or …
catalyzed multicomponent coupling and bis-cyclization have been developed. The mono-or …
Gold-catalyzed heteroannulation and allyl migration: synthesis of highly functionalized indole derivatives
KC Majumdar, S Hazra, B Roy - Tetrahedron letters, 2011 - Elsevier
Highly substituted indole derivatives have been prepared in good to excellent yields by a
novel gold-catalyzed cyclization accompanied by [3, 3]-migration of the allyl strategy. We …
novel gold-catalyzed cyclization accompanied by [3, 3]-migration of the allyl strategy. We …