[HTML][HTML] Gamma-aminobutyric acid and probiotics: Multiple health benefits and their future in the global functional food and nutraceuticals market

L Diez-Gutiérrez, L San Vicente, LJR Barrón… - Journal of Functional …, 2020 - Elsevier
Probiotics have attracted growing interest in recent decades due to their multiple health
benefits. The synergistic relationship between probiotics and prebiotics can enhance the …

GABAergic signaling by cells of the immune system: more the rule than the exception

AK Bhandage, A Barragan - Cellular and Molecular Life Sciences, 2021 - Springer
Gamma-aminobutyric acid (GABA) is best known as an essential neurotransmitter in the
evolved central nervous system (CNS) of vertebrates. However, GABA antedates the …

Neuroimmune pathophysiology in asthma

GF Pavón-Romero, NH Serrano-Pérez… - Frontiers in Cell and …, 2021 - frontiersin.org
Asthma is a chronic inflammation of lower airway disease, characterized by bronchial
hyperresponsiveness. Type I hypersensitivity underlies all atopic diseases including allergic …

Design and Synthesis of Novel Deuterated Ligands Functionally Selective for the γ-Aminobutyric Acid Type A Receptor (GABAAR) α6 Subtype with Improved …

DE Knutson, R Kodali, B Divović… - Journal of medicinal …, 2018 - ACS Publications
Recent reports indicate that α6β2/3γ2 GABAAR selective ligands may be important for the
treatment of trigeminal activation-related pain and neuropsychiatric disorders with sensori …

[HTML][HTML] Verification of Lactobacillus brevis tolerance to simulated gastric juice and the potential effects of postbiotic gamma-aminobutyric acid in streptozotocin …

A Abdelazez, H Abdelmotaal, SE Evivie… - Food Science and …, 2022 - Elsevier
The therapeutic effect of gamma-aminobutyric acid (GABA) on diabetes was spread as one
of the alarming epidemics worldwide. The study aims to investigate the function of …

A Novel Orally Available Asthma Drug Candidate That Reduces Smooth Muscle Constriction and Inflammation by Targeting GABAA Receptors in the Lung

GS Forkuo, AN Nieman, R Kodali, NM Zahn… - Molecular …, 2018 - ACS Publications
We describe lead compound MIDD0301 for the oral treatment of asthma based on
previously developed positive allosteric α5β3γ2 selective GABAA receptor (GABAAR) …

Design, synthesis, and biological evaluation of novel spiro imidazobenzodiazepines to identify improved inhaled bronchodilators

DA Webb, MJ Meyer, KM Medubi… - Journal of Medicinal …, 2023 - ACS Publications
Novel gamma-aminobutyric acid receptor (GABAAR) ligands structurally related to
imidazobenzodiazepine MIDD0301 were synthesized using spiro-amino acid N …

[HTML][HTML] GABAA receptor subtypes regulate stress-induced colon inflammation in mice

M Seifi, S Rodaway, U Rudolph, JD Swinny - Gastroenterology, 2018 - Elsevier
Background & Aims Psychological stress, in early life or adulthood, is a significant risk factor
for inflammatory disorders, including inflammatory bowel diseases. However, little is known …

Molecular characterization of GABA-A receptor subunit diversity within major peripheral organs and their plasticity in response to early life psychosocial stress

EA Everington, AG Gibbard, JD Swinny… - Frontiers in Molecular …, 2018 - frontiersin.org
Gamma aminobutyric acid (GABA) subtype A receptors (GABAARs) are integral membrane
ion channels composed of five individual proteins or subunits. Up to 19 different GABAAR …

Gut health benefits and associated systemic effects provided by functional components from the fermentation of natural matrices

R Colucci Cante, F Nigro, F Passannanti… - … Reviews in Food …, 2024 - Wiley Online Library
Recently, the role of the gut microbiota in metabolic health, immunity, behavioral balance,
longevity, and intestine comfort has been the object of several studies from scientific …