More than 60 years have passed since I. Ugi synthesized the first α-amidoamides in one
experimental step involving a combination of aldehydes, amines, carboxylic acids and …

The Ugi three component reaction (U‐3CR) is a variation of the famous Ugi reaction,
discovered almost 60 years ago. Today it is somehow neglected, compared to the classical …

A series of novel Benzofuran-tetrazole derivatives were successfully synthesised by
integrating multicomponent Ugi-azide reaction with the molecular hybridization approach …

We report the unprecedent Pd (I) catalyzed ring-opening arylation of cyclopropyl-α-
aminoamides. This protocol allows facile access to biologically important α-ketoamide …

Advances in base‐mediated post‐Ugi transformations are reported and discussed. The
minireview encompasses reports showing the abstraction of an alpha proton adjacent to …

The aerobic oxidative cleavage of Passerini and Ugi adducts in the presence of base and
copper (I) iodide is studied in detail. The oxidative cleavage yields α-ketoamides along with …

The deployment of multicomponent reactions (MCRs), defined as containing three or more
reactants, not only enjoys pot, atom, and step‐economy in the synthesis of novel complex …

Copper‐assisted post‐Ugi reactions enable access to different heterocyclic systems,
tetrahydronaphthoazetidinone, 2, 5‐dioxo‐1, 4‐methanobenzoazepine and 3 …

A facile multicomponent synthesis of novel thiazolidinone‐bis Schiff base hybrids has been
developed using readily available starting materials. The four‐component reaction of …

The successive treatment of aryl bromides with n-BuLi, DMF, hydroxylamine hydrochloride,
and finally diphenylphosphoryl azide provided efficiently the corresponding 5-aryltetrazoles …