The medicinal chemistry of piperazines: A review
The versatile basic structure of piperazine allows for the development and production of
newer bioactive molecules that can be used to treat a wide range of diseases. Piperazine …
newer bioactive molecules that can be used to treat a wide range of diseases. Piperazine …
Design, synthesis, α-amylase and glucose diffusion inhibition, and molecular docking studies of new indenopyrazolones bearing benzothiazole derivatives
R Punia, S Mor, S Sindhu, D Kumar, PP Das… - Bioorganic & Medicinal …, 2024 - Elsevier
An eco-friendly facile synthesis of a series of twenty 1-(4/6-substitutedbenzo [d] thiazol-2-yl)-
3-(phenyl/substitutedphenyl) indeno [1, 2-c] pyrazol-4 (1H)-ones 7a–t was achieved by the …
3-(phenyl/substitutedphenyl) indeno [1, 2-c] pyrazol-4 (1H)-ones 7a–t was achieved by the …
Synthesis, biological evaluation and mechanism of action of benzothiazole derivatives with aromatic hydrazone moiety, a new class of antileishmanial compounds
ES Coimbra, LMR Antinarelli… - Chemical Biology & …, 2024 - Wiley Online Library
Leishmaniasis is a disease caused by protozoa Leishmania spp., considered as a
significant and urgent public health problem mainly in developing countries. In the absence …
significant and urgent public health problem mainly in developing countries. In the absence …
COX inhibitory profiles of a series of thiadiazole-benzothiazole hybrids
A Özdemir, HE Temel - European Journal of Life Sciences, 2024 - dergipark.org.tr
In an endeavour to identify small molecule COX-1 inhibitors, a colorimetric assay protocol
was applied for the in vitro evaluation of COX-1 and 2 inhibitory potential of a series of …
was applied for the in vitro evaluation of COX-1 and 2 inhibitory potential of a series of …