Abstract α‐Aryl cyclocarbonyls are important building blocks in organic synthesis. While
many methods have been developed for their synthesis, the use of readily available and …

A catalyst-controlled divergent synthesis of bridged [3.3. 1] bis (indolyl)-oxanes and cis-[6.7]
fused bis (indolyl) oxepanes via diastereoselective desymmetrization of bis (indolyl) …

Reductive functionalization reactions between two electrophiles is a straightforward protocol
to access carbon‐carbon bonds without use of organometallic reagents prepared in …

An efficient method for the stereoselective synthesis of “all center substituted” polycyclic
pyrazoles from alkynyl cyclohexa-2, 5-dienones and nonstabilized diazoalkanes via …

An anion-relay double aza-Michael–Michael addition strategy has been reported for the
synthesis of intricate scaffolds from enone-tethered cyclohexadienones and primary amines …

An efficient functionalization of tyrosine residues in phenolic regions is achieved under
metal-free conditions. The strategy involves the conversion of a tyrosine residue to 4-amino …

Described herein is the development of an organoaluminium‐mediated tandem conjugate
addition‐cyclization sequence of p‐quinone monoacetals with 2‐siloxyphenyl Grignard …

An efficient strategy to afford pyrrolidine derivatised peptides through late-stage modification
of tyrosine-containing short peptides is presented. The metal-free dearomative strategy …

An efficient and concise synthesis of highly functionalized bridged coumarins has been
developed through a diastereoselective double Michael addition reaction of p‐quinols with …