Cellular senescence signaling in cancer: A novel therapeutic target to combat human malignancies

S Fakhri, SZ Moradi, LK DeLiberto… - Biochemical pharmacology, 2022 - Elsevier
Senescence is a special state of tumor suppression induced by cell cycle arrest. However,
releasing senescence-associated secretory phenotypes by senescent cells could provide …

[HTML][HTML] Chemoprevention curcumin analog 1.1 promotes metaphase arrest and enhances intracellular reactive oxygen species levels on TNBC MDA-MB-231 and …

D Novitasari, RI Jenie, J Kato… - Research in …, 2023 - journals.lww.com
Background and purpose: Previous studies highlighted that chemoprevention curcumin
analog-1.1 (CCA-1.1) demonstrated an antitumor effect on breast, leukemia, and colorectal …

Identification of potential targets of the curcumin analog CCA-1.1 for glioblastoma treatment: integrated computational analysis and in vitro study

A Hermawan, F Wulandari, N Hanif, RY Utomo… - Scientific Reports, 2022 - nature.com
The treatment of glioblastoma multiforme (GBM) is challenging owing to its localization in the
brain, the limited capacity of brain cells to repair, resistance to conventional therapy, and its …

Preparation and cytotoxic evaluation of PGV-1 derivative, CCA-1.1, as a new curcumin analog with improved-physicochemical and pharmacological properties

RY Utomo, F Wulandari, D Novitasari… - Advanced …, 2021 - pmc.ncbi.nlm.nih.gov
Purpose: This study aimed to challenge the anticancer potency of pentagamavunone-1
(PGV-1) and obtain a new compound (Chemoprevention-Curcumin Analog 1.1, CCA-1.1) …

[HTML][HTML] CCA-1.1, a novel curcumin analog, exerts cytotoxic anti-migratory activity toward TNBC and HER2-enriched breast cancer cells

D Novitasari, RI Jenie, RY Utomo, J Kato… - Asian Pacific Journal …, 2021 - ncbi.nlm.nih.gov
Objective: Chemoprevention curcumin Analog-1.1 (CCA-1.1) demonstrates antineoplastic
effect toward cancer cells. By using triple-negative breast cancer (TNBC), 4T1, and human …

[HTML][HTML] Tumour‐suppressive effects of curcumin analogs CCA‐1.1 and pentagamavunone‐1 in colon cancer: in vivo and in vitro studies

F Wulandari, M Ikawati, S Widyarini… - Journal of advanced …, 2023 - journals.lww.com
This study aimed to evaluate the efficacy of Chemoprevention Curcumin Analog-1.1 (CCA-
1.1) and Pentagamavunone-1 (PGV-1) in vivo and in vitro in colorectal cancer model. CCA …

Pentagamavunone-1 inhibits aggressive breast cancer cell proliferation through mitotic catastrophe and ROS-mediated activities: in vitro and in vivo studies

D Novitasari, I Nakamae, RI Jenie… - Saudi Pharmaceutical …, 2024 - Elsevier
Abstract Pentagamavunone-1 (PGV-1), an analog of curcumin, has been studied for its
cytotoxic effects in 4T1, MCF7, MCF7/HER2, and T47D breast cancer cells. Its …

PGV-1 permanently arrests HepG2 cells in M phase and inhibits liver carcinogenesis in DMH-induced rats

D Novitasari, J Kato, DDP Putri… - Journal of Applied …, 2023 - japsonline.com
Abstract Pentagamavunone-1 (PGV-1) has been reported to eliminate cancer cell
progression in the breast, blood, and colon. The current approach evaluates its …

A new curcumin analog, CCA-1.1, induces cell death and cell cycle arrest in WiDr colon cancer cells via ROS generation

F Wulandari, M Ikawati, M Kirihata, JY Kato… - Journal of Applied …, 2021 - japsonline.com
Abstract The new Pentagamavunone-1 (PGV-1) derivative, chemoprevention-curcumin
analog 1.1 (CCA-1.1), is described as an improved physicochemical feature with similar …

Africa leaf (Vernonia amygdalina Delille.) DCM extract synergistically supports growth suppression effect of doxorubicin on MCF7 and MCF7/HER2 with different …

NP Hapsari, DR Rahmawati, N Nugraheni… - Journal of Applied …, 2024 - japsonline.com
Africa leaf (Vernonia amygdalina Delille) has low cytotoxic activities against several cancer
cells. We evaluated its combination treatment with doxorubicin against luminal breast cancer …