Condensations of thioamides with acetylenecarboxylic acid derivatives

NA Danilkina, LE Mikhailov, BA Ivin - Russian journal of organic chemistry, 2006 - Springer
The review summarizes published data on the reactions of cyclic and acyclic thioamides
with derivatives of acetylenecarboxylic acids, which lead to the formation of both acyclic and …

Synergizing structure and function: cinnamoyl hydroxamic acids as potent urease inhibitors

LPS Viana, GM Naves, IG Medeiros, AS Guimarães… - Bioorganic …, 2024 - Elsevier
The current investigation encompasses the structural planning, synthesis, and evaluation of
the urease inhibitory activity of a series of molecular hybrids of hydroxamic acids and …

Regioselectivity of the alkylation of S-substituted 1,2,4-triazoles with dihaloalkanes

ATA Boraei, ESH El Ashry, A Duerkop - Chemistry Central Journal, 2016 - Springer
Abstract Background 1, 2, 4-Triazole3-thiones are good scaffolds for preparation of new lead
compounds. Their derivatives attracted the attention of chemists due to their wide spectrum …

Regioselective synthesis, characterization and antimicrobial evaluation of S-glycosides and S, N-diglycosides of 1, 2-Dihydro-5-(1H-indol-2-yl)-1, 2, 4-triazole-3-thione

H El Sayed, H El Sayed, MED Abd El Fattah… - European Journal of …, 2013 - Elsevier
Abstract Glycosylation of 1, 2-Dihydro-5-(1 H-indol-2-yl)-1, 2, 4-triazole-3-thione with 2, 3, 4,
6-tetra-O-acetyl-α-d-glucopyranosyl bromide, 2, 3, 4, 6-tetra-O-acetyl-α-d-galactopyranosyl …

Regioselective synthesis of new imidazo[4,5‐e][1,3]thiazino[2,3‐c][1,2,4]triazines via reaction of imidazo[4,5‐e][1,2,4]triazinethiones with ethyl phenylpropiolate

DB Vinogradov, AN Izmest'ev… - Journal of …, 2024 - Wiley Online Library
A method for the regioselective synthesis of imidazo [4, 5‐e][1, 3] thiazino [2, 3‐c][1, 2, 4]
triazine derivatives has been developed by the reaction of imidazotriazinethiones with ethyl …

[PDF][PDF] Chemistry of 1, 3-thiazin-4-ones and their derivatives, 1995-mid 2018

LJ Silverberg, QJ Moyer - Arkivoc, 2019 - researchgate.net
This review updates an earlier review published in 1996 by Ryabukhin, Korzhavina, and
Suzdalev, which covered the literature through 1994. It deals with the synthesis and …

Condensation of 5-(4-methylphenyl)-2,4-dihydro-3H-1,2,4-triazole-3-thione with haloacetic acids

AA Rzhevskii, NP Gerasimova, EM Alov… - Russian Chemical …, 2012 - Springer
Reactions of triazolethiones with haloacetic acids were studied with 5-(4-methylphenyl)-2, 4-
dihydro-3 H-1, 2, 4-triazole-3-thione as an example. It was proved for the first time by X-ray …

Cyclocondensation of N-aryl-3-oxobutanethioamides with 1H-1,2,4-triazol-5-amine

VN Britsun - Russian Journal of Organic Chemistry, 2008 - Springer
Abstract Reactions of N-aryl-3-oxobutanethioamides with 1 H-1, 2, 4-triazole-5-amine give
mixtures of 7-arylamino-5-methyl [1, 2, 4] triazolo [1, 5-a] pyrimidines, 5-methyl-4, 7-dihydro …

Ácidos cinamoilidroxâmicos como inibidores de urease: síntese, avaliação da atividade inibitória e estudos sobre o mecanismo de inibição

LPS Viana - 2024 - repositorio.ufmg.br
Os ácidos hidroxâmicos (AHs) compõem uma classe de compostos reconhecida pelas suas
propriedades quelantes e capacidade de inibir importantes metaloenzimas contendo Ni (II) …

Reaction of 3-oxo-N-phenylbutanethioamide with 5-amino-1H-1,2,4-triazoles

VN Britsun, AN Borisevich, LS Samoilenko… - Russian journal of …, 2006 - Springer
Abstract Reactions of 3-oxo-N-phenylbutanethioamide with 3-substituted 5-amino-1 H-1, 2,
4-triazoles in acetic acid led to the formation of 5-methyl-7, 8-dihydro [1, 2, 4] triazolo [1, 5-a] …