N-Acylsulfonamides strongly inhibit human carbonic anhydrase isoenzymes I and II
Sulfonamides represent a significant class of biologically active compounds that inhibit
carbonic anhydrase (CA, EC.: 4.2. 1.1) isoenzymes involved in different pathological and …
carbonic anhydrase (CA, EC.: 4.2. 1.1) isoenzymes involved in different pathological and …
The synthesis of unsubstituted cyclic imides using hydroxylamine under microwave irradiation
E Benjamin, Y Hijji - Molecules, 2008 - mdpi.com
Unsubstituted cyclic imides were synthesized from a series of cyclic anhydrides,
hydroxylamine hydrochloride (NH2OH∙ HCl), and 4-N, N-dimethylamino-pyridine (DMAP …
hydroxylamine hydrochloride (NH2OH∙ HCl), and 4-N, N-dimethylamino-pyridine (DMAP …
[PDF][PDF] Efficient microwave assisted syntheses of unsubstituted cyclic imides
YMBE Hijji, E Benjamin - Heterocycles, 2006 - triggered.edina.clockss.org
A number of cyclic imides were synthesized from cyclic anhydrides using ammonium
chloride (NH4Cl), and 4-N, N-dimethylaminopyridine (DMAP) or with ammonium acetate …
chloride (NH4Cl), and 4-N, N-dimethylaminopyridine (DMAP) or with ammonium acetate …
A novel bioactive compounds of 2-azetidinone derived from pyrazin dicarboxylic acid: synthesis and antmicrobial screening
AN Ayyash, HQA Habeeb - ACTA Pharmaceutica Sciencia, 2019 - actapharmsci.com
ABSTRACT A series of novel 2-azetidinons entitled N, N'-bis [3-chloro-2-oxo-4-(substituted
pyridine-2-yl)-azetidin-1-yl] pyrazine-2, 3-dicarboxamide and N, N'-bis [3, 3-dichloro-2-oxo-4 …
pyridine-2-yl)-azetidin-1-yl] pyrazine-2, 3-dicarboxamide and N, N'-bis [3, 3-dichloro-2-oxo-4 …
Synthesis of N-unsubstituted cyclic imides from anhydride with urea in deep eutectic solvent (DES) choline chloride/urea
L Liu, HY Zhang, G Yin, Y Zhang, J Zhao - Chemical Papers, 2020 - Springer
N-Unsubstituted cyclic imides were readily synthesized in deep eutectic solvent (DES)
choline chloride (ChCl)/urea from anhydrides with urea. Urea serves as both a DES …
choline chloride (ChCl)/urea from anhydrides with urea. Urea serves as both a DES …
[PDF][PDF] Microwave-promoted synthesis of cyclic imides.
IA Perillo, MS Shmidt, SC Prieto… - ARKIVOC: Online Journal …, 2018 - arkat-usa.org
Cyclic imides have been extensively investigated because of the wide range of biological
activities they exert, as well as due to their importance as synthetic intermediates …
activities they exert, as well as due to their importance as synthetic intermediates …
Synthesis of Some New Pyrrolo[3,4-f]isoindole Derivatives Bearing a 1,3-Thiazolidin-4-one Moiety
AN Ayyash, DK Kafi, YK Jabur - Russian Journal of Organic Chemistry, 2022 - Springer
A series of new N, N′-bis [4-oxo-2-(pyridine-2-yl)-1, 3-thiazolidin-3-yl]-2, 2′-[1, 3, 5, 7-
tetraoxo-5, 7-dihydropyrrolo [3, 4-f] isoindole-2, 6 (1 H, 3 H)-diyl] diacetamide derivatives …
tetraoxo-5, 7-dihydropyrrolo [3, 4-f] isoindole-2, 6 (1 H, 3 H)-diyl] diacetamide derivatives …
Synthesis and Antimicrobial Screening of Novel Azetidin-2-ones Derived from Pyromellitic Diimide via [2+ 2]-Cycloaddition Reaction
AN Ayyash - Russian Journal of Organic Chemistry, 2019 - Springer
A series of novel 2-azetidinone derivatives have been obtained starting from pyromellitic
dianhydride. Pyromellitic dianhydride was converted to pyromellitic diimide using sodium …
dianhydride. Pyromellitic dianhydride was converted to pyromellitic diimide using sodium …
[PDF][PDF] Diels-Alder reaction of 2-(cyclic amino)-substituted 3-furancarbonitriles with maleimides to phthalimides
H Maruoka, F Okabe, Y Koutake… - …, 2009 - triggered.stanford.clockss.org
An efficient Diels-Alder reaction is described in the furan series, leading to phthalimides in
high yields. Thermal treatment of 2-(4-morpholinyl, 1-piperidinyl, and 1-pyrrolidinyl)-3 …
high yields. Thermal treatment of 2-(4-morpholinyl, 1-piperidinyl, and 1-pyrrolidinyl)-3 …
[HTML][HTML] Full Text HTML
H Maruoka, F Okabe, Y Koutake, T Fujioka… - triggered.edina.clockss.org
An approach to dihydroindoles and tetrahydroquinolines from N-alkenylated 2-acylamino-3-
furancarbonitriles via a [4+ 2] cycloaddition reaction is described. Thermal treatment of N …
furancarbonitriles via a [4+ 2] cycloaddition reaction is described. Thermal treatment of N …