Artificial intelligence to deep learning: machine intelligence approach for drug discovery

R Gupta, D Srivastava, M Sahu, S Tiwari, RK Ambasta… - Molecular …, 2021 - Springer
Drug designing and development is an important area of research for pharmaceutical
companies and chemical scientists. However, low efficacy, off-target delivery, time …

AI in drug discovery and its clinical relevance

R Qureshi, M Irfan, TM Gondal, S Khan, J Wu, MU Hadi… - Heliyon, 2023 - cell.com
The COVID-19 pandemic has emphasized the need for novel drug discovery process.
However, the journey from conceptualizing a drug to its eventual implementation in clinical …

Learning functional properties of proteins with language models

S Unsal, H Atas, M Albayrak, K Turhan… - Nature Machine …, 2022 - nature.com
Data-centric approaches have been used to develop predictive methods for elucidating
uncharacterized properties of proteins; however, studies indicate that these methods should …

Advances in de novo drug design: from conventional to machine learning methods

VD Mouchlis, A Afantitis, A Serra, M Fratello… - International journal of …, 2021 - mdpi.com
De novo drug design is a computational approach that generates novel molecular structures
from atomic building blocks with no a priori relationships. Conventional methods include …

Deep learning in virtual screening: recent applications and developments

TB Kimber, Y Chen, A Volkamer - International journal of molecular …, 2021 - mdpi.com
Drug discovery is a cost and time-intensive process that is often assisted by computational
methods, such as virtual screening, to speed up and guide the design of new compounds …

Comprehensive survey of recent drug discovery using deep learning

J Kim, S Park, D Min, W Kim - International Journal of Molecular Sciences, 2021 - mdpi.com
Drug discovery based on artificial intelligence has been in the spotlight recently as it
significantly reduces the time and cost required for developing novel drugs. With the …

Drug–target affinity prediction using graph neural network and contact maps

M Jiang, Z Li, S Zhang, S Wang, X Wang, Q Yuan… - RSC …, 2020 - pubs.rsc.org
Computer-aided drug design uses high-performance computers to simulate the tasks in drug
design, which is a promising research area. Drug–target affinity (DTA) prediction is the most …

Artificial intelligence in drug discovery: applications and techniques

J Deng, Z Yang, I Ojima, D Samaras… - Briefings in …, 2022 - academic.oup.com
Artificial intelligence (AI) has been transforming the practice of drug discovery in the past
decade. Various AI techniques have been used in many drug discovery applications, such …

FP-GNN: a versatile deep learning architecture for enhanced molecular property prediction

H Cai, H Zhang, D Zhao, J Wu… - Briefings in …, 2022 - academic.oup.com
Accurate prediction of molecular properties, such as physicochemical and bioactive
properties, as well as ADME/T (absorption, distribution, metabolism, excretion and toxicity) …

Geometric interaction graph neural network for predicting protein–ligand binding affinities from 3d structures (gign)

Z Yang, W Zhong, Q Lv, T Dong… - The journal of physical …, 2023 - ACS Publications
Predicting protein–ligand binding affinities (PLAs) is a core problem in drug discovery.
Recent advances have shown great potential in applying machine learning (ML) for PLA …