Synthesis, biological evaluation, and docking studies of 3-(substituted)-aryl-5-(9-methyl-3-carbazole)-1H-2-pyrazolines as potent anti-inflammatory and antioxidant …
A novel series of 3-(substituted)-aryl-5-(9-methyl-3-carbazole)-1H-2-pyrazolines (5a–o) has
been synthesized and the structures of newly synthesized compounds were characterized …
been synthesized and the structures of newly synthesized compounds were characterized …
Valorization of onion solid waste and their flavonols for assessment of cytotoxicity, enzyme inhibitory and antioxidant activities
Onion (Allium cepa L.) is rich with flavonols which perceived benefits to human health.
Flavonols like quercetin and quercetin glycosides from onion solid waste (OSW) have been …
Flavonols like quercetin and quercetin glycosides from onion solid waste (OSW) have been …
Synthesis of extended conjugated indolyl chalcones as potent anti-breast cancer, anti-inflammatory and antioxidant agents
PS Bhale, HV Chavan, SB Dongare… - Bioorganic & medicinal …, 2017 - Elsevier
In the present investigation, synthesis of a series of extended conjugated δ-chloro-α-cyano
substituted indolyl chalcones (5a–p) was accomplished by reacting 3-cyanoacetylindole 2 …
substituted indolyl chalcones (5a–p) was accomplished by reacting 3-cyanoacetylindole 2 …
Inhibition properties of propolis extracts to some clinically important enzymes
The present study was conducted to envisage inhibition effects of propolis on the crucial
enzymes, urease, xanthine oxidase (XO) and acetylcholinesterase (AChE). Some of the …
enzymes, urease, xanthine oxidase (XO) and acetylcholinesterase (AChE). Some of the …
Honey as an apitherapic product: its inhibitory effect on urease and xanthine oxidase
H Sahin - Journal of enzyme inhibition and medicinal chemistry, 2016 - Taylor & Francis
The aim of this study was to evaluate new natural inhibitor sources for the enzymes urease
and xanthine oxidase (XO). Chestnut, oak and polyfloral honey extracts were used to …
and xanthine oxidase (XO). Chestnut, oak and polyfloral honey extracts were used to …
Heterocyclic curcumin derivatives of pharmacological interest: Recent progress
M Martinez-Cifuentes, B Weiss-Lopez… - Current Topics in …, 2015 - ingentaconnect.com
Curcumin, a natural yellow polyphenol, is isolated from the herb Curcuma longa L.(turmeric),
a member of the ginger family. It has been extensively studied due to their multiple …
a member of the ginger family. It has been extensively studied due to their multiple …
Synthesis and pharmacological evaluation of combretastatin-A4 analogs of pyrazoline and pyridine derivatives as anticancer, anti-inflammatory and antioxidant …
SN Shringare, HV Chavan, PS Bhale… - Medicinal Chemistry …, 2018 - Springer
Three category of N 1-phenyl pyrazoline (5a–e), N 1-phenyl-sulfonyl pyrazoline (6a–e), and
pyridine analogs (8a–d) of combretastatin-A4 were synthesized. The structures of …
pyridine analogs (8a–d) of combretastatin-A4 were synthesized. The structures of …
Synthesis and pharmacological evaluation of pyrazoline and pyrimidine analogs of combretastatin-A4 as anticancer, anti-inflammatory and antioxidant agents
SN Shringare, HV Chavan, PS Bhale… - Croatica Chemica …, 2018 - hrcak.srce.hr
Sažetak A library of 3, 5-diaryl-1-carbothioamide-pyrazoline (5a–j), N1-phenyl sulfonyl
pyrazoline (6a–e) and pyrimidine (7a) analogs of combretastatin-A4 were synthesized and …
pyrazoline (6a–e) and pyrimidine (7a) analogs of combretastatin-A4 were synthesized and …
PEG Mediated Synthesis and Biological Evaluation of Asymmetrical Pyrazole Curcumin Analogues as Potential Analgesic, Anti‐Inflammatory and Antioxidant Agents
SY Jadhav, RB Bhosale, SP Shirame… - Chemical Biology & …, 2015 - Wiley Online Library
The new series of asymmetrical pyrazole curcumin analogues 4a–g were synthesized by
using polyethylene glycol (PEG‐400) as a green reaction medium and evaluated for their in …
using polyethylene glycol (PEG‐400) as a green reaction medium and evaluated for their in …
Synthesis and biological evaluation of novel series of aminopyrimidine derivatives as urease inhibitors and antimicrobial agents
A novel series of carbazole substituted aminopyrimidines (5a-p) were synthesized and
screened for their in vitro urease inhibition and antimicrobial activity. Among the compounds …
screened for their in vitro urease inhibition and antimicrobial activity. Among the compounds …