Weak Nucleophiles in the Aza‐Michael Reaction

AY Rulev - Advanced Synthesis & Catalysis, 2023 - Wiley Online Library
Abstract The 1, 4‐conjugated addition of nitrogen centered nucleophiles to electron‐
deficient alkenes is one of the most significant and widely used reactions in modern …

Asymmetric organocatalytic approach to 2, 4-disubstituted 1, 2, 3-triazoles by N2-selective aza-Michael addition

UK Bhagat, RK Peddinti - The Journal of organic chemistry, 2018 - ACS Publications
Despite the fact that N1-functionalization of NH-1, 2, 3-triazoles has been known for several
decades, enantioselective variants of this reaction have only recently been developed …

Silver-Catalyzed Cascade Cyclization of Amino-NH-1,2,3-Triazoles with 2-Alkynylbenzaldehydes: An Access to Pentacyclic Fused Triazoles

S Zhang, J Li, T Xiao, B Yang, Y Jiang - Molecules, 2022 - mdpi.com
An operationally simple Ag (I)-catalyzed approach for the synthesis of isoquinoline and
quinazoline fused 1, 2, 3-triazoles was developed by a condensation and amination …

Synthesis of Highly Substituted 1, 2, 4-Triazole-Based 3-Nitrochromanes through Aza-Michael Addition Reaction under Catalyst-and Base-Free Conditions

T Das, SP Parida, S Mohapatra, S Nayak - Synthesis, 2024 - thieme-connect.com
A simple and efficient aza-Michael addition reaction of 1, 2, 4-triazoles to functionalized 2-
aryl-3-nitro-2H-chromenes has been demonstrated under catalyst-and base-free conditions …

An FeCl 3-catalyzed three-component reaction for the synthesis of β-(1, 2, 3-triazolyl)-ketones using DMF as a one-carbon source

R Fang, L Zheng, X Chen, C Wang… - Organic & Biomolecular …, 2024 - pubs.rsc.org
An FeCl3-catalyzed oxidative condensation of NH-1, 2, 3-triazoles, aryl methyl ketones (or
acetophenones) and DMF (N, N-dimethylformamide) for the synthesis of β-(1, 2, 3-triazolyl) …

The versatility of DABCO: synthetic applications of its basic, nucleophilic, and catalytic properties Part 2*. Catalysis of Michael and Biginelli reactions and nucleophilic …

DI Bugaenko, AV Karchava, MA Yurovskaya - Chemistry of Heterocyclic …, 2020 - Springer
The versatility of DABCO: synthetic applications of its basic, nucleophilic, and catalytic
properties Part 2*. Catalysis of Michael and Biginelli reactions and nucleophilic addition at C=X …

Lithium Chloride Catalyzed Aza-Michael Addition of Pyrazoles to α, β-Unsaturated Imides

H Zhou, X Xiang, B Ma, G Wang, Z Zhang, J Yang - Synthesis, 2019 - thieme-connect.com
A lithium chloride catalyzed aza-Michael reaction of pyrazoles to α, β-unsaturated imides
has been developed. A range of aromatic and aliphatic α, β-unsaturated imides are found to …

4-单取代-1, 2, 3-三氮唑的修饰转化研究进展

杨保民, 张水滔, 董鲜, 秦贵平, 江玉波 - 化学学报, 2023 - sioc-journal.cn
摘要1, 2, 3-三氮唑是一类广泛应用在医药, 农药以及材料等领域的五元氮杂环结构. 自2002
年Sharpless 和Meldal 等发展了铜催化叠氮-炔偶极环加成反应以来, 1, 2, 3 …

Catalyst‐Free Selective Aza‐Michael Addition of 3‐Aminopyrazole to Nitroalkenes

Z Li, W Song - ChemistrySelect, 2018 - Wiley Online Library
Catalyst‐free N1 selective aza‐Michael addition of 3‐aminopyrazole to nitroalkenes is
described. A series of 1‐(2‐nitro‐1‐arylethyl)‐1H‐pyrazol‐3‐amines were efficiently …

Five-membered ring systems: with more than one N atom

L Yet - Progress in Heterocyclic Chemistry, 2020 - Elsevier
Five-Membered Ring Systems: With More than One N Atom - ScienceDirect Skip to main
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