A comprehensive account on recent progress in pharmacological activities of benzimidazole derivatives

SR Brishty, MJ Hossain, MU Khandaker… - Frontiers in …, 2021 - frontiersin.org
Nowadays, nitrogenous heterocyclic molecules have attracted a great deal of interest
among medicinal chemists. Among these potential heterocyclic drugs, benzimidazole …

Aminobenzimidazoles and Structural Isomers as Templates for Dual‐Acting Butyrylcholinesterase Inhibitors and hCB2R Ligands To Combat Neurodegenerative …

D Dolles, M Nimczick, M Scheiner, J Ramler… - …, 2016 - Wiley Online Library
A pharmacophore model for butyrylcholinesterase (BChE) inhibitors was applied to a human
cannabinoid subtype 2 receptor (hCB2R) agonist and verified it as a first‐generation lead for …

Synthesis, binding assays, cytotoxic activity and docking studies of benzimidazole and benzothiophene derivatives with selective affinity for the CB2 cannabinoid …

J Romero-Parra, J Mella-Raipán, V Palmieri… - European Journal of …, 2016 - Elsevier
Herein we report the design, synthesis, bioinformatic and biological studies of
benzimidazole and benzothiophene derivatives as new cannabinoid receptor ligands. To …

Combined CoMFA and CoMSIA 3D-QSAR study of benzimidazole and benzothiophene derivatives with selective affinity for the CB2 cannabinoid receptor

J Romero-Parra, H Chung, RA Tapia… - European Journal of …, 2017 - Elsevier
The preceding years have brought an exponential increase in our understanding of the
endocannabinoid system (ECS), including the knowledge of CB1 and CB2 cannabinoid …

Impact of Cannabinoid Receptors in the Design of Therapeutic Agents against Human Ailments

A Kumar, O Gupta, R Bhatia… - Current Topics in …, 2023 - benthamdirect.com
The Cannabinoid (CB) signalling cascade is widely located in the human body and is
associated with several pathophysiological processes. The endocannabinoid system …

Motifs in Natural Products as Useful Scaffolds to Obtain Novel Benzo[d]imidazole-Based Cannabinoid Type 2 (CB2) Receptor Agonists

AYH Cho, H Chung, J Romero-Parra, P Kumar… - International Journal of …, 2023 - mdpi.com
The endocannabinoid system (ECS) constitutes a broad-spectrum modulator of homeostasis
in mammals, providing therapeutic opportunities for several pathologies. Its two main …

Computational Modeling of Non-active Functional States of the Cannabinoid Receptor 1 and its Ligands

AO Aderibigbe - 2021 - search.proquest.com
Abstract The cannabinoid receptor 1 (CB1) is a class A G-protein coupled receptor that is
implicated in a variety of physiological processes, such as energy homeostasis, appetite …

Búsqueda De Moduladores Del Sistema Endocannabinoide: Síntesis Y Evaluación Biológica De Carbamoilos De Anillos Benzoimidazólicos, Diseñados Por …

RAE Valderrama - 2021 - search.proquest.com
Desde tiempos remotos, la Cannabis ha sido utilizada tanto por sus acciones medicinales
como por sus efectos recreacionales. En la actualidad, hay un sin número de estudios …

[引用][C] Búsqueda de moduladores del sistema endocannabinoide: síntesis y evaluación biológica de carbamoilos de anillos benzoimidazólicos, diseñados por …

RA Escobar Valderrama - 2021

[引用][C] El patrimonio en la recuperación de Santiago nor-poniente: Barrio Portales

JI Tapia - 2007 - Pontificia Universidad Católica de …