Synthesis and antiviral evaluation of some sugar arylglycinoylhydrazones and their oxadiazoline derivatives

MT Abdel‐Aal, WA El‐Sayed… - Archiv der Pharmazie …, 2006 - Wiley Online Library
Abstract Sugar N‐arylaminoacetylhydrazones 2–5 were prepared by the reaction of N‐
arylaminoacetylhydrazides 1 with equivalent amounts of the corresponding …

Acyclonucleosides: part 1. seco-Nucleosides

ESH El Ashry, Y El Kilany - Advances in heterocyclic chemistry, 1996 - Elsevier
This chapter is the first of a sequence of three chapters that will appear in successive
volumes of this series dealing with the chemistry of acyclonucleosides. Acyclonucleosides …

[PDF][PDF] Tandem in situ generation and 1, 5-electrocyclization of N-hetaryl nitrilimines. A facile methodology for synthesis of annulated 1, 2, 4-triazoles and their acyclo C …

AS Shawali - Arkivoc, 2010 - arkat-usa.org
This review summarizes results of literature reports concerning tandem in situ generation
and 1, 5-electrocyclization of N-hetaryl nitrilimines reported by us and other research groups …

Synthesis and antiviral evaluation of sugar uracil-1-ylmethylhydrazones and their oxadiazoline derivatives

OM Ali, HH Amer, AH Adel - Synthesis, 2007 - thieme-connect.com
Carbethoxymethyluracils have been synthesized and derivatized to the corresponding
hydrazides, which were reacted with monosaccharides to afford the corresponding sugar …

Acyclo C-Nucleoside Analogs. Regioselective Annellation of a Triazole Ring to 5-Methyl-1,2,4-Triazino[5,6-b]Indole and Formation of Certain 3-Poly Hydroxyalkyl …

N Rashed, HA Hamid, ES Ramadan… - Nucleosides & …, 1998 - Taylor & Francis
Cyclodehydrogenation of the ethylidene derivative of (5-methyl-1, 2, 4-triazino [5, 6-b] indol-
3-yl) hydrazine (1) gave the angular isomer, 1, 10-dimethyl-1, 2, 4-triazolo [3′, 4′: 3, 4][1 …

Syntheses and in silico pharmacokinetic predictions of glycosylhydrazinyl-pyrazolo [1, 5-c] pyrimidines and pyrazolo [1, 5-c] triazolo [4, 3-a] pyrimidines as anti …

KFM Atta, OOM Farahat, TQ Al-Shargabi… - Medicinal Chemistry …, 2019 - Springer
Abstract New glycosylhydrazinyl-pyrazolo [1, 5-c] pyrimidines were synthesized by the
reaction of respective 5-aryl-7-hydrazino-2-phenylpyrazolo [1, 5-c] pyrimidines (1a-d) with …

Synthesis of acyclo C-nucleosides of phenanthro [9, 10-e][1, 2, 4] triazino [3, 4-c]-[1, 2, 4] triazoles, and their precursors

A Hamed, ER Abo-Amaym… - Nucleosides & …, 1998 - Taylor & Francis
ABSTRACT Reaction of 3-hydrazinophenanthro [9, 10-e][1, 2, 4] triazine (1) with aliphatic
and aromatic aldehydes as well as monosaccharides gave the corresponding hydrazones …

Synthesis and Dimroth Rearrangement of 6-Cyano-l, 2, 4-triazolo-[4, 3-a] pyrimidin-5-and 7-ones. A Novel Alkylation with Orthoesters and a New Participation of the …

ESH El Ashry, Y El Kilany, N Rashed… - … für Naturforschung B, 1998 - degruyter.com
The cyclization products of 5-cyano-2-hydrazino-6-phenyl-3, 4-dihydropyrimidin-4-one (6)
with one carbon inserting agents have been confirmed to be of the 1, 2, 4-triazolo [4, 3-a] …

Synthesis of hydantoin nucleosides with naphthylmethylene substituents in the 5-position

AI Khodair, ESE Ibrahimb - Nucleosides, Nucleotides & Nucleic …, 1996 - Taylor & Francis
Abstract (Z)-5-(Naphthylmethylene)-2-thiohydantoin derivatives (3a, b, 12a-d) were
prepared directly fiom condensations of 2-thiohydantoin derivatives (1, l la, b) with …

Acyclo C-nucleosides analogues of condensed 1, 2, 4-triazines

ESH El Ashry, N Rashed, HA Hamid… - … für Naturforschung B, 1997 - degruyter.com
Acyclo C-nucleosides of 7-methyl-10H-1, 2, 4-triazolo [3', 4': 3, 4][1, 2, 4] triazino [5, 6-b]
indoles (9) have been prepared by cyclodehydrogenation of the sugar derivatives of 3 …