Development of new antimycobacterial sulfonyl hydrazones and 4-methyl-1, 2, 3-thiadiazole-based hydrazone derivatives
VT Angelova, T Pencheva, N Vassilev, E K-Yovkova… - Antibiotics, 2022 - mdpi.com
Fifteen 4-methyl-1, 2, 3-thiadiazole-based hydrazone derivatives 3a–d and sulfonyl
hydrazones 5a–k were synthesized. They were characterized by 1H-NMR, 13C NMR, and …
hydrazones 5a–k were synthesized. They were characterized by 1H-NMR, 13C NMR, and …
[HTML][HTML] Synthesis of hydrazides of heterocyclic amines and their antimicrobial and spasmolytic activity
DA Berillo, MA Dyusebaeva - Saudi Pharmaceutical Journal, 2022 - Elsevier
Un unsolvable issue of a significant number increase of drug multi resistant strains of
microorganisms including Mycobacterium tuberculosis force researchers for continuous …
microorganisms including Mycobacterium tuberculosis force researchers for continuous …
Bioactive sulfonyl hydrazones with alkyl derivative: Characterization, ADME properties, molecular docking studies and investigation of inhibition on choline esterase …
In this work, new sulfonylhydrazone compounds with alkyl derivatives (SH1–SH4 series)
were synthesized via a green chemistry method, and their inhibition effects on …
were synthesized via a green chemistry method, and their inhibition effects on …
Designing heterocyclic chalcones, benzoyl/sulfonyl hydrazones: An insight into their biological activities and molecular docking study
The aim of this study is to investigate the antioxidant, anticholinesterase and the
antiproliferative activities of some chalcones, benzoyl and sulfonyl hydrazones. The …
antiproliferative activities of some chalcones, benzoyl and sulfonyl hydrazones. The …
New piperidine-hydrazone derivatives: Synthesis, biological evaluations and molecular docking studies as AChE and BChE inhibitors
Hydrazones and the piperidine ring containing compounds were considered as beneficial
substrates in drug design. Therefore, this study was aimed at the synthesis of new benzoyl …
substrates in drug design. Therefore, this study was aimed at the synthesis of new benzoyl …
Synthesis of arylsulfonyl hydrazone derivatives: antioxidant activity, acetylcholinesterase inhibition properties, and molecular docking study
In this current paper, fifteen novel sulfonyl hydrazone derivatives have been successfully
synthesized and evaluated for antioxidant activity as well as their effects on inhibitory activity …
synthesized and evaluated for antioxidant activity as well as their effects on inhibitory activity …
Synthesis, crystal structure, hirshfeld surface analysis and computational study of hydrazone derivative of 5, 5-dimethylcyclohexane-1, 3-dione
M Kurbanova, M Ashfaq, A Sadigova… - Journal of Structural …, 2023 - Springer
The diazotization reaction of p-fluoroaniline from aromatic amines with 5, 5-
dimethylcyclohexane-1, 3-dione was studied, as a result 2-(2-(p-fluorophenyl) hydrazone)-5 …
dimethylcyclohexane-1, 3-dione was studied, as a result 2-(2-(p-fluorophenyl) hydrazone)-5 …
Synthesis of benzoyl hydrazones having 4-hydroxy-3, 5-dimethoxy phenyl ring, theirbiological activities, and molecular modeling studies on enzyme inhibition …
Hydrazone compounds have high capacity in terms of antioxidant activity and enzyme
inhibition activities such as anticholinesterase, tyrosinase, and urease. In this study, benzoyl …
inhibition activities such as anticholinesterase, tyrosinase, and urease. In this study, benzoyl …
Synthesis, Antioxidant and Some Enzyme Inhibition Activities of New Sulfonyl Hydrazones and their Molecular Docking Simulations
In this work, a series of new sulfonyl hydrazones were synthesized and screened for
antioxidant and anticholinesterase, tyrosinase and urease enzyme inhibition activities. In …
antioxidant and anticholinesterase, tyrosinase and urease enzyme inhibition activities. In …
Exploring novel nitrofuranyl sulfonohydrazides as anti‐Leishmania and anti‐cancer agents: Synthesis, in vitro efficacy and hit identification
C Kannigadu, J Aucamp… - Chemical Biology & Drug …, 2022 - Wiley Online Library
Leishmaniasis and cancer are two deadly diseases that plague the human population.
There are a limited number of drugs available for the treatment of these diseases; however …
There are a limited number of drugs available for the treatment of these diseases; however …