Structural Perspective into Thiazoles and other Azole Derivatives as Anthelmintic Agents

M Vajedpour, JA Shiran, A Ashnamoghadam… - Acta Tropica, 2024 - Elsevier
Helminths or worm-like parasites are common infectious pathogens that cause significant
diseases and mortality in animals and humans. To be noted, nematodes or soil-transmitted …

[HTML][HTML] Synthetic approaches and biological evaluation of nitrogen bridgehead thiazolo [3, 2-a] pyrimidines

M Abdel-Megid, KM El-mahdy, AM Elkazak, SE Zarif… - Results in …, 2024 - Elsevier
Thiazolopyrimidines are bicyclic compounds formed by the fusion of thiazole and pyrimidine
rings in a single molecular frame. The fusion of these two heterocyclic systems containing …

[PDF][PDF] Green expedient synthesis of pyrimidine derivatives via chalcones and evaluation of their anthelmintic activity

BM Sahoo, M Rajeswari… - Indian Journal of …, 2017 - pdfs.semanticscholar.org
Objective: In the present study, we focused on the environment-friendly processes used for
the preparation of pyrimidine derivatives with pharmacological properties. In this regard …

Synthesis and anticancer activity evaluation of novel azacalix [2] arene [2] pyrimidines

Y Addepalli, X Yang, M Zhou, DP Reddy… - European journal of …, 2018 - Elsevier
A series of novel azacalix [2] arene [2] pyrimidines were synthesized, and evaluated for their
antiproliferative activities against A549, MCF7, SH-SY5Y and CNE human cancer cell lines …

Synthesis, structural characterization and DFT study of N-(pyrimidyl)-ω-amino acids/peptide: β-alanine, γ-aminobutyric acid, 5-aminovaleric acid, 6-aminohexanoic …

A García-Raso, A Terrón, JJ Fiol, A López-Zafra… - …, 2023 - pubs.rsc.org
In this manuscript we report the synthesis and structural characterization of five pyrimidine
amino acid/peptide modified derivatives: N-(2-pyrimidyl)-β-alanine (pyr-β-Ala)(1), N-(2 …

Virtual Analysis of Condensed Pyrimidine Derivatives as COX II Inhibitors Potential Anti-inflammatory Agents

SA Khedkar, JS Patil, PM Sabale - Research Journal of …, 2021 - indianjournals.com
Drug design and development is an interactive process includes process like molecular
docking which involves virtual analysis of the derivatives against the protein targets. COXS …

Modified-amino acid/peptide pyrimidine analogs: synthesis, structural characterization and DFT studies of N-(pyrimidyl) gabapentine and N-(pyrimidyl) baclofen

A García-Raso, A Terrón, JJ Fiol… - New Journal of …, 2021 - pubs.rsc.org
In this manuscript, we report the synthesis and structural characterization of two new
pyrimidine amino acid modified derivatives: N-(pyrimidyl) gabapentin (pyr-gabapentin)(1) …

[PDF][PDF] Detailed CV

MSM Phil - Chemistry, 2002 - mangaloreuniversity.ac.in
Detailed CV Name: Dr. RAMESH SABU GANI Educational Qualification: M.Sc. M.Phil. Ph.D.
Designation: Assistant Professor Address f Page 1 Detailed CV Name: Dr. RAMESH SABU …