Recent studies of nitrogen and sulfur containing heterocyclic analogues as novel antidiabetic agents: a review
S Gharge, SG Alegaon - Chemistry & Biodiversity, 2024 - Wiley Online Library
The prevalence of diabetes mellitus is on the rise, which demands the identification of novel
antidiabetic drugs. There is a need for safer and more effective alternatives because the …
antidiabetic drugs. There is a need for safer and more effective alternatives because the …
2-Aminobenzothiazoles in anticancer drug design and discovery
G Huang, T Cierpicki, J Grembecka - Bioorganic chemistry, 2023 - Elsevier
Cancer is one of the major causes of mortality and morbidity worldwide. Substantial
research efforts have been made to develop new chemical entities with improved anticancer …
research efforts have been made to develop new chemical entities with improved anticancer …
Multifunctional catalysis of nanosheet defective molybdenum sulfide basal planes for tandem reactions involving alcohols and molecular hydrogen
M Rodenes, F Dhaeyere, S Martín… - ACS Sustainable …, 2023 - ACS Publications
Establishing tandem catalytic synthetic strategies based on the use of readily available,
stable, and renewable feedstocks is of great significant for the sustainable advancement of …
stable, and renewable feedstocks is of great significant for the sustainable advancement of …
An ROS-Responsive Donor That Self-Reports Its H2S Delivery by Forming a Benzoxazole-Based Fluorophore
Hydrogen sulfide (H2S), an endogenous signaling molecule, is known to play a pivotal role
in neuroprotection, vasodilation, and hormonal regulation. To further explore the biological …
in neuroprotection, vasodilation, and hormonal regulation. To further explore the biological …
Assessment of the inhibitory efficacy of a thiazole derivative as an efficient corrosion inhibitor for augmenting the resistance of MS in acidic environments
Numerous thiazole compounds have been developed as cutting-edge inhibitors because of
a rising fascination with using corrosion inhibitors (CIs) and preventative measures to …
a rising fascination with using corrosion inhibitors (CIs) and preventative measures to …
A β-ketoenamine-linked covalent organic framework as a heterogeneous photocatalyst for the synthesis of 2-arylbenzothiazoles by cyclization reaction
Z Liu, Z Chen, H Tong, M Ji, W Chu - Green Chemistry, 2023 - pubs.rsc.org
Visible light-mediated catalysis has gradually become an important means of green catalytic
organic synthesis. However, traditional photosensitizers (organic dyes or precious transition …
organic synthesis. However, traditional photosensitizers (organic dyes or precious transition …
Advances in the discovery of heterocyclic-based drugs against Alzheimer's disease
Introduction Alzheimer's disease is a multifactorial neurodegenerative disorder
characterized by beta-amyloid accumulation and tau protein hyperphosphorylation. The …
characterized by beta-amyloid accumulation and tau protein hyperphosphorylation. The …
Advances in chalcone derivatives: Unravelling their anticancer potential through structure-activity studies
KA Sheikh, A Gupta, M Umar, R Ali… - Journal of Molecular …, 2024 - Elsevier
Cancer continues to be a global health challenge, thereby necessitating the evolution of
innovative therapeutic strategies. The synthesis of chalcone derivatives has garnered …
innovative therapeutic strategies. The synthesis of chalcone derivatives has garnered …
Benzothiazole a privileged scaffold for Cutting-Edges anticancer agents: Exploring drug design, structure-activity relationship, and docking studies
Cancer is a major societal, public health, and economic burden in the 21 st century, with 9.7
million deaths in 2022 (9.96 million in 2020) and 20 million new cancer cases (19.6 million …
million deaths in 2022 (9.96 million in 2020) and 20 million new cancer cases (19.6 million …
A General C–N Cross-Coupling to Synthesize Heteroaryl Amines Using a Palladacyclic N-Heterocyclic Carbene Precatalyst
R Fan, M Kuai, D Lin, F Bauer, W Fang - Organic Letters, 2022 - ACS Publications
A new palladacyclic N-heterocyclic carbene precatalyst was designed by the combination of
1, 3-bis (2, 6-diisopropylphenyl) acenaphthoimidazol-2-ylidene (AnIPr) with an achiral 2 …
1, 3-bis (2, 6-diisopropylphenyl) acenaphthoimidazol-2-ylidene (AnIPr) with an achiral 2 …