Carbazole 1 was isolated first from coal tar in 1872 by Graebe and Glazer (Figure 1). 1 In
1965, Chakraborty et al. described the isolation and antibiotic properties of murrayanine …

Upon reaction with IPy2BF4, 4-substituted anilines give regioselectively the corresponding o-
iodoanilines in nearly quantitative yield, in a process that can be carried out on a multigram …

Synthetic melatonin was iodinated by treatment with potassium iodide in the presence of an
oxidizing agent, Iodo-Gen. The iodination products of melatonin were extracted with …

The first hydroboration of an 1-alkynylamide—the electronically modulated variant of an
ynamine—is described. This hydroboration in combination with a Suzuki–Miyaura cross …

Structural diversity in heterocyclic chemistry is key to unlocking new properties and modes of
action. In this regard, heterocycles embedding emerging fluorinated substituents hold great …

Highly regioselective synthesis of 2,4,5-(hetero)aryl substituted oxazoles by intermolecular [3+2]-cycloaddition
of unsymmetrical internal alkynes - Chemical Communications (RSC Publishing) DOI:10.1039/C3CC45410J …

The Nazarov cyclization of divinyl ketones gives access to cyclopentenones. Replacing one
of the vinyl groups by a cyclopropane leads to a formal homo‐Nazarov process for the …

The human antigen R (HuR) is an RNA-binding protein known to modulate the expression of
target mRNA coding for proteins involved in inflammation, tumorigenesis, and stress …

The highly stereoselective asymmetric 6π-azaelectrocyclization was achieved as a general
synthetic method based on the reaction between the (E)-3-carbonyl-2, 4, 6-trienal …

The word indole is derived from the word India: indigo (3), the blue dye, was first exported
from India to Europe in the 16th century. Indoles are generally crystalline colorless solids …