Pyridazinic bioisosteres with potential applications in medicinal chemistry and agriculture
RA Tucaliuc, V Mangalagiu, II Mangalagiu - Processes, 2023 - mdpi.com
Bioisosteres are substituents or groups (atoms, ions, or molecules) with similar chemical or
physical properties, and which usually have similar biological properties. Pyridazine and its …
physical properties, and which usually have similar biological properties. Pyridazine and its …
Benzoquinoline derivatives: A straightforward and efficient route to antibacterial and antifungal agents
V Antoci, L Oniciuc, D Amariucai-Mantu… - Pharmaceuticals, 2021 - mdpi.com
We report here the design, synthesis, experimental and in silico evaluation of the
antibacterial and antifungal activity of some new benzo [f] quinoline derivatives. Two classes …
antibacterial and antifungal activity of some new benzo [f] quinoline derivatives. Two classes …
Hybrids Diazine: Recent Advancements in Modern Antimicrobial Therapy
Nowadays, antimicrobial therapies have become a very challenging issue because of a
large diversity of reasons such as antimicrobial resistance, over consumption and misuse of …
large diversity of reasons such as antimicrobial resistance, over consumption and misuse of …
Norlabdane compounds containing thiosemicarbazone or 1, 3-thiazole fragments: Synthesis and antimicrobial activity
New di-, tri-, tetra-, and pentanorlabdane compounds with thiosemicarbazone and 1, 3-
thiazole fragments were synthesized. Their antifungal and antibacterial activities were …
thiazole fragments were synthesized. Their antifungal and antibacterial activities were …
Discovery of a Biocontrol Strain Trichaptum laricinum: Its Metabolites and Antifungal Activity against Pathogenic Fungus Colletotrichum anthrisci
SS Huang, HX Yang, J He, JK Liu… - Journal of Agricultural …, 2024 - ACS Publications
Finding safe and environmentally friendly fungicides is one of the important strategies in
modern pesticide research and development. In this work, the antipathogenic effects of the …
modern pesticide research and development. In this work, the antipathogenic effects of the …
Synthesis and evaluation of biological activity of homodrimane sesquiterpenoids bearing 1, 3, 4-oxadiazole or 1, 3, 4-thiadiazole units
L Lungu, A Ciocarlan, C Smigon, I Ozer… - Chemistry of …, 2020 - Springer
Synthesis of novel (+)-sclareolide-based homodrimane sesquiterpenoids bearing 1, 3, 4-
oxadiazole or 1, 3, 4-thiadiazole units has been reported. These terpeno-heterocyclic …
oxadiazole or 1, 3, 4-thiadiazole units has been reported. These terpeno-heterocyclic …
Synthesis of new homodrimane sesquiterpenoids containing diazine, 1, 2, 4-triazole and carbazole rings
The present paper reports on six step synthesis of 11-homodrim-6, 8-dien-12-oic acid N-
substituted amides containing diazine, 1, 2, 4-triazole and carbazole rings based on …
substituted amides containing diazine, 1, 2, 4-triazole and carbazole rings based on …
Hybrid Quinoline-Sulfonamide Complexes (M2+) Derivatives with Antimicrobial Activity
D Diaconu, V Mangalagiu, D Amariucai-Mantu… - Molecules, 2020 - mdpi.com
Two new series of hybrid quinoline-sulfonamide complexes (M2+: Zn2+, Cu2+, Co2+ and
Cd2+) derivatives (QSC) were designed, synthesized and tested for their antimicrobial …
Cd2+) derivatives (QSC) were designed, synthesized and tested for their antimicrobial …
Synthesis and Antimicrobial Activity Evaluation of Homodrimane Sesquiterpenoids with a Benzimidazole Unit
Herein we report a feasible study concerning the synthesis and the in vitro antimicrobial
activity of some new homodrimane sesquiterpenoids with a benzimidazole unit. Based on …
activity of some new homodrimane sesquiterpenoids with a benzimidazole unit. Based on …
Synthesis of homodrimane sesquiterpenoids bearing 1, 3-benzothiazole unit and their antimicrobial activity evaluation
Based on some homodrimane carboxylic acids and their acyl chlorides, a series of fourteen
2-homodrimenyl-1, 3-benzothiazoles, N-homodrimenoyl-2-amino-1, 3-benzothiazoles, 4 …
2-homodrimenyl-1, 3-benzothiazoles, N-homodrimenoyl-2-amino-1, 3-benzothiazoles, 4 …