Sulfonimidamides: synthesis and applications in preparative organic chemistry

GC Nandi, PI Arvidsson - Advanced synthesis & catalysis, 2018 - Wiley Online Library
During the last one and half decades, chemists within vastly different areas of science have
witnessed a rising interest in chemical matters incorporating the sulfonimidamide functional …

Synthesis of amino-functionalized sulfonimidamides and their application in the enantioselective Henry reaction

M Steurer, C Bolm - The Journal of Organic Chemistry, 2010 - ACS Publications
Amino-functionalized sulfonimidamides have been prepared by aziridinium ring-opening
reactions and nucleophilic substitutions of sulfonimidoyl chlorides. Whereas the former …

Discovery of N-Cyano-sulfoximineurea Derivatives as Potent and Orally Bioavailable NLRP3 Inflammasome Inhibitors

S Agarwal, S Sasane, HA Shah… - ACS medicinal …, 2020 - ACS Publications
NLRP3 inflammasome mediated release of interleukin-1β (IL-1β) has been implicated in
various diseases. In this study, rationally designed mimics of sulfonylurea moiety were …

Synthesis of CF3-Substituted Sulfoximines from Sulfonimidoyl Fluorides

R Kowalczyk, AJF Edmunds, RG Hall, C Bolm - Organic Letters, 2011 - ACS Publications
N-Protected trifluoromethyl-substituted sulfoximines have been prepared by treatment of
sulfonimidoyl fluorides with a combination of the Ruppert− Prakash reagent (TMSCF3) and …

Syntheses and Transformations of sulfinamides

Q Zhang, J Xi, H Ze, Z Qingle - Synthesis, 2021 - thieme-connect.com
Sulfinamides, especially enantiopure sulfinamides, are widely used in organic and
medicinal synthesis. Syntheses and transformations of racemic and enantioenriched …

Synthesis of Enantiopure Sulfonimidamides and Elucidation of Their Absolute Configuration by Comparison of Measured and Calculated CD Spectra and X‐Ray …

C Worch, I Atodiresei, G Raabe… - Chemistry–A European …, 2010 - Wiley Online Library
Straightforward syntheses of enantiopure N‐benzoyl‐and N‐tert‐butyloxycarbonyl‐
protected sulfonimidamides, which can be used as building blocks in newly designed …

Regioselective Chlorothiolation of Alkenes with Sulfonyl Chlorides

J Wei, S Liang, L Jiang, Y Mumtaz… - The Journal of Organic …, 2019 - ACS Publications
Newly developed sulfonyl chloride-based regioselective chlorothiolation of alkenes has
been disclosed; the reaction is compatible with a variety of functional groups and can be …

Trimorphism of an asymmetric disulfonamide Schiff base

J Sanmartín, F Novio, AM García-Deibe… - New Journal of …, 2007 - pubs.rsc.org
An asymmetric Schiff base, H2L, has been prepared by condensation of the selectively
functionalised 2-(tosylaminomethyl) aniline (A) with 2-tosylaminobenzaldehyde (B). H2L has …

The use of two optically active N-sulfinyl α-imino esters in the stereoselective aza-Diels–Alder reaction

T Andreassen, M Lorentzen, LK Hansen, OR Gautun - Tetrahedron, 2009 - Elsevier
Diastereoselective aza-Diels–Alder (aza-DA) reactions of ethyl (S)-N-(tert-butanesulfinyl)
iminoacetate (2a) and ethyl (S)-N-(p-toluenesulfinyl) iminoacetate (2b) with different dienes …

[图书][B] Handbook of reagents for organic synthesis: Reagents for heteroarene synthesis

AB Charette - 2017 - books.google.com
The Handbook is a compilation of 99 articles on diverse reagents and catalysts that describe
the synthesis of heteroarenes, the building blocks of a wide range of chemicals used in …